CENTRAL SEROTONIN-LIKE ACTIVITY OF "6-CHLORO-2-[1-PIPERAZINYL]-PYRAZINE (CPP-MK-212)

被引:51
作者
CLINESCHMIDT, BV [1 ]
MCGUFFIN, JC [1 ]
PFLUEGER, AB [1 ]
机构
[1] MERCK INST THERAPEUT RES,W POINT,PA 19486
关键词
D O I
10.1016/0014-2999(77)90117-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:65 / 74
页数:10
相关论文
共 28 条
[1]  
Anden N E, 1968, Adv Pharmacol, V6, P347
[2]  
ANDEN NE, 1970, INT S AMPHETAMINES R, P447
[3]   ANTAGONISM OF 5-HYDROXYTRYPTAMINE-INDUCED BRONCHOSPASM IN GUINEA-PIGS BY 8BETA-CARBOBENZYLOXYAMINOMETHYL-1-METHYL-10ALPHA-ERGOLINE [J].
BERETTA, C ;
GLASSER, AH ;
NOBILI, MB ;
SILVESTR.R .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1965, 17 (07) :423-&
[4]   MODEL FOR QUANTITATIVE STUDY OF CENTRAL DOPAMINERGIC AND SEROTONINERGIC ACTIVITY [J].
BIEGER, D ;
HORNYKIEWICZ, O ;
LAROCHELLE, L .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1972, 18 (01) :128-+
[5]   ROLE OF MONOAMINES IN ANOREXIGENIC ACTIONS OF FENFLURAMINE, AMPHETAMINE AND PARA-CHLOROMETHAMPHETAMINE [J].
CLINESCHMIDT, BV ;
MCGUFFIN, JC ;
WERNER, AB .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1974, 27 (03) :313-323
[6]   INDOLEAMINE ANTAGONISTS - RELATIVE POTENCIES AS INHIBITORS OF TRYPTAMINE-EVOKED EVOKED AND 5-HYDROXYTRYPTOPHAN-EVOKED RESPONSES [J].
CLINESCHMIDT, BV ;
LOTTI, VJ .
BRITISH JOURNAL OF PHARMACOLOGY, 1974, 50 (02) :311-313
[7]   CENTRAL CATECHOLAMINE RECEPTOR BLOCKING ACTIONS OF BE-2254 (HEAT) - COMPARISON WITH CHLORPROMAZINE AND HALOPERIDOL [J].
CLINESCHMIT, BV ;
PFLUEGER, AB ;
BUNTING, PR ;
MCGUFFIN, JC ;
BALLENTINE, RJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1975, 32 (02) :279-286
[8]   NEW PERIPHERAL ANTAGONISTS OF 5-HYDROXYTRYPTAMINE [J].
COPP, FC ;
GREEN, AF ;
HODSON, HF ;
RANDALL, AW ;
SIM, MF .
NATURE, 1967, 214 (5084) :200-&
[9]   A METHOD FOR ASSESSING EFFECTS OF DRUGS ON CENTRAL ACTIONS OF 5-HYDROXYTRYPTAMINE [J].
CORNE, SJ ;
WARNER, BT ;
PICKERING, RW .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1963, 20 (01) :106-&
[10]   ROLE OF RAPHE AND EXTRAPYRAMIDAL NUCLEI IN STEREOTYPED AND CIRCLING RESPONSES TO QUIPAZINE [J].
COSTALL, B ;
NAYLOR, RJ .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1975, 27 (05) :368-371