PROPOSED DOPAMINERGIC PHARMACOPHORE OF LERGOTRILE, PERGOLIDE, AND RELATED ERGOT ALKALOID DERIVATIVES

被引：72

作者：

CANNON, JG ^{[1
]}

DEMOPOULOS, BJ ^{[1
]}

LONG, JP ^{[1
]}

FLYNN, JR ^{[1
]}

SHARABI, FM ^{[1
]}

机构：

[1] UNIV IOWA,COLL MED,DEPT PHARMACOL,IOWA CITY,IA 52242

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1981年 / 24卷 / 03期

关键词：

D O I：

10.1021/jm00135a002

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：238 / 240

页数：3

共 24 条

[1] BICYCLIC AND TRICYCLIC ERGOLINE PARTIAL STRUCTURES - RIGID 3-(2-AMINOETHYL)PYRROLES AND 3-(2-AMINOETHYL)PYRAZOLE AND 4-(2-AMINOETHYL)PYRAZOLE AS DOPAMINE AGONISTS [J].

BACH, NJ ;

KORNFELD, EC ;

JONES, ND ;

CHANEY, MO ;

DORMAN, DE ;

PASCHAL, JW ;

CLEMENS, JA ;

SMALSTIG, EB .

JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (05) :481-491

[2] CONVERSION OF ERGOLINES TO HEXAHYDROBENZO[F]QUINOLINES AND OCTAHYDROBENZO[F]QUINOLINES (DEPYRROLOERGOLINES) [J].

BACH, NJ ;

KORNFELD, EC ;

CLEMENS, JA ;

SMALSTIG, EB .

JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (07) :812-814

[3]

BACH NJ, 1978, Patent No. 4110339

[4]

Cannon J G, 1975, Adv Neurol, V9, P177

[5] CENTRALLY ACTING EMETICS 10 RIGID DOPAMINE CONGENERS DERIVED FROM OCTAHYDROBENZO[F]QUINOLINE [J].

CANNON, JG ;

HATHEWAY, GJ ;

LONG, JP ;

SHARABI, FM .

JOURNAL OF MEDICINAL CHEMISTRY, 1976, 19 (08) :987-993

[6]

CANNON JG, 1979, PERIPHERAL DOPAMINER, P87

[7]

FINNEY DJ, 1952, STATISTICAL METHODS, P139

[8] EFFECTS OF (8-BETA)-8-[(METHYLTHIO)METHYL]-6-PROPYLERGOLINE ON DOPAMINERGIC FUNCTION AND BRAIN DOPAMINE TURNOVER IN RATS [J].

FULLER, RW ;

CLEMENS, JA ;

KORNFELD, EC ;

SNODDY, HD ;

SMALSTIG, EB ;

BACH, NJ .

LIFE SCIENCES, 1979, 24 (04) :375-382

[9] 3-[2-(DIPROPYLAMINO)ETHYL]PHENOL - NEW AND SELECTIVE DOPAMINERGIC AGENT [J].

GEISSLER, HE .

ARCHIV DER PHARMAZIE, 1977, 310 (09) :749-756

[10] COMPARISON OF VASCULAR DOPAMINE RECEPTOR WITH OTHER DOPAMINE RECEPTORS [J].

GOLDBERG, LI ;

VOLKMAN, PH ;

KOHLI, JD .

ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1978, 18 :57-79

← 1 2 3 →