METHYLENE PIPERAZINE-2,5-DIONES AS TEMPLATES FOR THE SYNTHESIS OF AMINO-ACID DERIVATIVES

被引：27

作者：

CHAI, CLL ^{[1
]}

KING, AR ^{[1
]}

机构：

[1] AUSTRALIAN NATL UNIV,THE FACULTIES,DEPT CHEM,CANBERRA,ACT 0200,AUSTRALIA

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 24期

关键词：

D O I：

10.1016/0040-4039(95)00743-V

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Methylene piperazine-2,5-diones 5a and 5b are important synthetic intermediates. The preparation as well as the use of these compounds in the synthesis of amino acid derivatives are described. Our studies demonstrate that excellent chiral induction in carbon-carbon bond forming reactions can be obtained with methylene piperazinedione 5b.

引用

页码：4295 / 4298

页数：4

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