SYNTHESES OF HETEROCYCLES .135. QUINOLIZINES AND INDOLIZINES .6. A SYNTHESIS OF 2-HYDROXY-4H-BENZO[A]QUINOLIZIN-4-ONES

被引：10

作者：

KAPPE, T

LINNAU, Y

机构：

[1] Institut für Organische Chemie der Universität Graz, Graz

来源：

MONATSHEFTE FUR CHEMIE | 1969年 / 100卷 / 05期

关键词：

D O I：

10.1007/BF00900194

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The condensation of 1-alkyl-3.4-dihydro-isoquinolines (1a to g) with 2.4.6-trichlorophenyl malonates (2a-e) yields 2-hydroxy-6,7-dihydro-4 H-benzo[a]quinolizin-4-ones (3a-p). Yields, required reaction-periods and temperatures are depending on the nature of the substituents present in the malonyl and isoquinoline residue. © 1969 Springer-Verlag.

引用

页码：1726 / &

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