IS STIMULATION OF BENZODIAZEPINE RECEPTOR-BINDING MEDIATED BY A NOVEL GABA RECEPTOR

被引:134
作者
KAROBATH, M [1 ]
PLACHETA, P [1 ]
LIPPITSCH, M [1 ]
LARSEN, PK [1 ]
机构
[1] ROYAL DANISH SCH PHARM, DEPT CHEM BC, DK-2100 COPENHAGEN, DENMARK
关键词
D O I
10.1038/278748a0
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
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页码:748 / 749
页数:2
相关论文
共 15 条
[1]   NEW CONCEPTS ON MECHANISM OF ACTION OF BENZODIAZEPINES [J].
COSTA, E ;
GUIDOTTI, A ;
MAO, CC ;
SURIA, A .
LIFE SCIENCES, 1975, 17 (02) :167-185
[2]   PROPERTIES OF GAMMA-AMINOBUTYRIC ACID (GABA) RECEPTOR-BINDING IN RAT-BRAIN SYNAPTIC MEMBRANE-FRACTIONS [J].
ENNA, SJ ;
SNYDER, SH .
BRAIN RESEARCH, 1975, 100 (01) :81-97
[3]   ENDOGENOUS PROTEIN MODULATES AFFINITY OF GABA AND BENZODIAZEPINE RECEPTORS IN RAT-BRAIN [J].
GUIDOTTI, A ;
TOFFANO, G ;
COSTA, E .
NATURE, 1978, 275 (5680) :553-555
[4]  
Haefely W, 1975, Adv Biochem Psychopharmacol, P131
[5]   BETEL NUT CONSTITUENTS AS INHIBITORS OF GAMMA-AMINOBUTYRIC ACID UPTAKE [J].
JOHNSTON, GAR ;
KROGSGAARDLARSEN, P ;
STEPHANSON, A .
NATURE, 1975, 258 (5536) :625-628
[6]  
KAROBATH M, P NATN ACAD SCI US
[7]   INHIBITION OF GABA UPTAKE IN RAT-BRAIN SLICES BY NIPECOTIC ACID, VARIOUS ISOXAZOLES AND RELATED COMPOUNDS [J].
KROGSGAARDLARSEN, P ;
JOHNSTON, GAR .
JOURNAL OF NEUROCHEMISTRY, 1975, 25 (06) :797-802
[8]   STRUCTURE-ACTIVITY STUDIES ON INHIBITION OF GABA BINDING TO RAT-BRAIN MEMBRANES BY MUSCIMOL AND RELATED COMPOUNDS [J].
KROGSGAARDLARSEN, P ;
JOHNSTON, GAR .
JOURNAL OF NEUROCHEMISTRY, 1978, 30 (06) :1377-1382
[9]   FACILITATION OF BENZODIAZEPINE BINDING BY SODIUM-CHLORIDE AND GABA [J].
MARTIN, IL ;
CANDY, JM .
NEUROPHARMACOLOGY, 1978, 17 (11) :993-998
[10]   BENZODIAZEPINE RECEPTOR - DEMONSTRATION IN CENTRAL NERVOUS-SYSTEM [J].
MOHLER, H ;
OKADA, T .
SCIENCE, 1977, 198 (4319) :849-851