DIASTEREOSPECIFIC SYNTHESIS OF D-ALLO-THREONINE AND L-ALLO-THREONINE AND TRICHLORINATED DERIVATIVES SUITABLE FOR THE PREPARATION OF TRITIUM LABELED MATERIAL

被引：27

作者：

BEAULIEU, PL

机构：

[1] Bio-Méga Inc., Laval, Que. H7S 2G5

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 08期

关键词：

D O I：

10.1016/S0040-4039(00)74479-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

D- or L- serine can be converted to L- or D-gamma,gamma,gamma-trichloro-allo-threonine, which on catalytic hydrogenolysis give diastereomerically pure L-allo- or D-allo-threonine respectively. This procedure can be adapted to the preparation of tritium labelled material.

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页码：1031 / 1034

页数：4

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