SYNTHESIS OF 1-ALPHA,25-DIHYDROXY-22-THIAVITAMIN D-3 AND RELATED ANALOGS

被引：6
作者：
KAWASE, A [1 ]
HIRATA, M [1 ]
ENDO, K [1 ]
KUBODERA, N [1 ]
机构：
[1] CHUGAI PHARMACEUT CO LTD,FUJI GOTEMBA RES LABS,GOTEMBA,SHIZUOKA 412,JAPAN
来源：
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1995年 / 5卷 / 03期
关键词：
D O I：
10.1016/0960-894X(95)00015-L
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
The 22-thiolation reaction of the steroidal side chain and the synthesis of 1 alpha,25-dihydroxy-22-thiavitamin D-3 and related analogs bearing side chains of different sizes in combination with 20-epi configuration are described.
引用
收藏
页码：279 / 282
页数：4
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