IRAZEPINE, A NONCOMPETITIVE, IRREVERSIBLE INHIBITOR OF DIAZEPAM-H-3 BINDING TO BENZODIAZEPINE RECEPTORS

被引:41
作者
RICE, KC
BROSSI, A
TALLMAN, J
PAUL, SM
SKOLNICK, P
机构
[1] NIAMDD,BIOORGAN CHEM LAB,BETHESDA,MD 20014
[2] NIMH,BIOL PSYCHIAT BRANCH,BETHESDA,MD 20014
[3] NIMH,CLIN PSYCHOBIOL BRANCH,BETHESDA,MD 20014
关键词
D O I
10.1038/278854a0
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:854 / 855
页数:2
相关论文
共 19 条
[1]  
ASANO T, P NATN ACAD SCI US
[2]  
Assony S.J., 1961, ORGANIC SULFUR COMPO, P326, DOI [10.1016/B978-1-4831-9982-5.50031-2, DOI 10.1016/B978-1-4831-9982-5.50031-2]
[3]   BENZODIAZEPINE RECEPTORS - LABELING IN INTACT ANIMALS WITH [H-3]FLUNITRAZEPAM [J].
CHANG, RSL ;
SNYDER, SH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 48 (02) :213-218
[4]  
LIPPA A, PHARMAC BIOCH BEHAV
[5]  
MACDONALD JR, UNPUBLISHED
[6]   DEMONSTRATION OF AN ENDOGENOUS, COMPETITIVE INHIBITOR(S) OF [H-3] DIAZEPAM BINDING IN BOVINE BRAIN [J].
MARANGOS, PJ ;
PAUL, SM ;
GREENLAW, P ;
GOODWIN, FK ;
SKOLNICK, P .
LIFE SCIENCES, 1978, 22 (21) :1893-1900
[7]   PROPERTIES OF DIAZEPAM-H-3 BINDING TO BENZODIAZEPINE RECEPTORS IN RAT CEREBRAL-CORTEX [J].
MOHLER, H ;
OKADA, T .
LIFE SCIENCES, 1977, 20 (12) :2101-2110
[8]   BENZODIAZEPINE RECEPTOR - DEMONSTRATION IN CENTRAL NERVOUS-SYSTEM [J].
MOHLER, H ;
OKADA, T .
SCIENCE, 1977, 198 (4319) :849-851
[9]   RAPID CHANGES IN BRAIN BENZODIAZEPINE RECEPTORS AFTER EXPERIMENTAL SEIZURES [J].
PAUL, SM ;
SKOLNICK, P .
SCIENCE, 1978, 202 (4370) :892-894
[10]  
SEGEL IH, 1976, BIOCH CALCULATIONS, P256