A REDUCTIVE AMINATION/LACTAMIZATION PROCEDURE USING BOROHYDRIDE REAGENTS

被引：1

作者：

ABDELMAGID, AF

HARRIS, BD

MARYANOFF, CA

机构：

来源：

SYNLETT | 1994年 / 01期

关键词：

LACTAMIZATION; REDUCTIVE AMINATION; SODIUM TRIACETOXYBOROHYDRIDE; IMINE FORMATION; SODIUM BOROHYDRIDE;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

We report a procedure for tandem reductive amination-lactamization of aldehydes or ketones with aminoesters or ketoesters with primary amines under mild conditions (NaBH(OAc)(3)/1,2-dichloroethane or NaBH4/MeOH).

引用

页码：81 / 83

页数：3

共 15 条

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