CHARACTERIZATION OF THE INHIBITION OF U46619-MEDIATED HUMAN-PLATELET ACTIVATION BY THE TRIMETOQUINOL ISOMERS - EVIDENCE FOR ENDOPEROXIDE THROMBOXANE-A2 RECEPTOR BLOCKADE

被引:0
作者
AHN, CH
ROMSTEDT, KJ
WALLACE, LJ
MILLER, DD
FELLER, DR
机构
[1] OHIO STATE UNIV,COLL PHARM,DIV PHARMACOL,COLUMBUS,OH 43210
[2] OHIO STATE UNIV,COLL PHARM,DIV MED CHEM,COLUMBUS,OH 43210
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D O I
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中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:3023 / 3033
页数:11
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共 43 条
[1]   ENZYMATIC BASIS FOR PLATELET-AGGREGATION AND RELEASE - SIGNIFICANCE OF PLATELET-ATMOSPHERE AND RELATIONSHIP BETWEEN PLATELET-FUNCTION AND BLOOD-COAGULATION [J].
ARDLIE, NG ;
HAN, P .
BRITISH JOURNAL OF HAEMATOLOGY, 1974, 26 (03) :331-356
[2]   LIGAND-BINDING TO THROMBOXANE RECEPTORS ON HUMAN-PLATELETS - CORRELATION WITH BIOLOGICAL-ACTIVITY [J].
ARMSTRONG, RA ;
JONES, RL ;
WILSON, NH .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 79 (04) :953-964
[3]   PLATELET SEQUESTRATION IN MAN .1. METHODS [J].
ASTER, RH ;
JANDL, JH .
JOURNAL OF CLINICAL INVESTIGATION, 1964, 43 (05) :843-&
[4]   EFFECTS OF EPOXYMETHANO ANALOGS OF PROSTAGLANDIN ENDOPEROXIDES ON AGGREGATION, ON RELEASE OF 5-HYDROXYTRYPTAMINE AND ON THE METABOLISM OF 3',5'-CYCLIC-AMP AND CYCLIC-GMP IN HUMAN-PLATELETS [J].
BEST, LC ;
MCGUIRE, MB ;
MARTIN, TJ ;
PRESTON, FE ;
RUSSELL, RGG .
BIOCHIMICA ET BIOPHYSICA ACTA, 1979, 583 (03) :344-351
[5]  
BILLAH MM, 1982, J BIOL CHEM, V257, P1856
[6]   THE CYCLIC AMP-LOWERING EFFECT OF THE STABLE ENDOPEROXIDE ANALOG U46619 IN HUMAN-PLATELETS [J].
BONNE, C ;
MARTIN, B ;
REGNAULT, F .
THROMBOSIS RESEARCH, 1980, 20 (5-6) :701-704
[7]   AGGREGATION OF BLOOD PLATELETS BY ADENOSINE DIPHOSPHATE AND ITS REVERSAL [J].
BORN, GVR .
NATURE, 1962, 194 (4832) :927-&
[8]   PHOSPHATIDYLINOSITOL 4,5-BISPHOSPHATE MAY REPRESENT THE SITE OF RELEASE OF PLASMA MEMBRANE-BOUND CALCIUM UPON STIMULATION OF HUMAN-PLATELETS [J].
BROEKMAN, MJ .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 120 (01) :226-231
[9]   PHOSPHOLIPID-METABOLISM IN STIMULATED HUMAN-PLATELETS - CHANGES IN PHOSPHATIDYLINOSITOL, PHOSPHATIDIC-ACID, AND LYSOPHOSPHOLIPIDS [J].
BROEKMAN, MJ ;
WARD, JW ;
MARCUS, AJ .
JOURNAL OF CLINICAL INVESTIGATION, 1980, 66 (02) :275-283
[10]  
CASTAGNA M, 1982, J BIOL CHEM, V257, P7847