EFFECTS OF 1,3-DIPROPYL-8-CYCLOPENTYLXANTHINE (DPCPX), A HIGHLY SELECTIVE ADENOSINE RECEPTOR ANTAGONIST, ON FORCE OF CONTRACTION IN GUINEA-PIG ATRIAL AND VENTRICULAR CARDIAC PREPARATIONS

被引:46
作者
VONDERLEYEN, H
SCHMITZ, W
SCHOLZ, H
SCHOLZ, J
LOHSE, MJ
SCHWABE, U
机构
[1] UNIV HAMBURG,KRANKENHAUS EPPENDORF,ALLGEMEINE ABT,MARTINISTR 52,D-2000 HAMBURG 20,FED REP GER
[2] UNIV HEIDELBERG,INST PHARMAKOL,D-6900 HEIDELBERG,FED REP GER
关键词
D O I
10.1007/BF00168970
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:204 / 209
页数:6
相关论文
共 42 条
[1]  
BAER HP, 1985, ADENOSINE RECEPTORS, P247
[2]   AN IMPROVED ASSAY OF CYCLIC 3',5'-NUCLEOTIDE PHOSPHODIESTERASES WITH QAE-SEPHADEX COLUMNS [J].
BAUER, AC ;
SCHWABE, U .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1980, 311 (02) :193-198
[3]   ANTI-ADRENERGIC ACTION OF ADENOSINE ON VENTRICULAR MYOCARDIUM IN EMBRYONIC CHICK HEARTS [J].
BELARDINELLI, L ;
VOGEL, S ;
LINDEN, J ;
BERNE, RM .
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 1982, 14 (05) :291-294
[4]   ISOLATED ATRIAL MYOCYTES - ADENOSINE AND ACETYLCHOLINE INCREASE POTASSIUM CONDUCTANCE [J].
BELARDINELLI, L ;
ISENBERG, G .
AMERICAN JOURNAL OF PHYSIOLOGY, 1983, 244 (05) :H734-H737
[5]   MECHANISM OF ACTION AND CARDIOTONIC ACTIVITY OF A NEW PHOSPHODIESTERASE INHIBITOR, THE BENZIMIDAZOLE DERIVATIVE ADIBENDAN (BM 14.478), IN GUINEA-PIG HEARTS [J].
BETHKE, T ;
BRUNKHORST, D ;
VANDERLEYEN, H ;
MEYER, W ;
NIGBUR, R ;
SCHOLZ, H .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1988, 337 (05) :576-582
[6]   EVIDENCE FOR ADENOSINE RECEPTOR-MEDIATED ISOPRENALINE-ANTAGONISTIC EFFECTS OF THE ADENOSINE-ANALOGS PIA AND NECA ON FORCE OF CONTRACTION IN GUINEA-PIG ATRIAL AND VENTRICULAR CARDIAC PREPARATIONS [J].
BOHM, M ;
BRUCKNER, R ;
MEYER, W ;
NOSE, M ;
SCHMITZ, W ;
SCHOLZ, H ;
STARBATTY, J .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1985, 331 (2-3) :131-139
[7]   ROLE OF GUANINE NUCLEOTIDE-BINDING PROTEIN IN THE REGULATION BY ADENOSINE OF CARDIAC POTASSIUM CONDUCTANCE AND FORCE OF CONTRACTION - EVALUATION WITH PERTUSSIS TOXIN [J].
BOHM, M ;
BRUCKNER, R ;
NEUMANN, J ;
SCHMITZ, W ;
SCHOLZ, H ;
STARBATTY, J .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1986, 332 (04) :403-405
[8]  
BOHM M, 1984, J PHARMACOL EXP THER, V230, P483
[9]   CARDIAC EFFECT OF ADENOSINE - MECHANISM OF ACTION, PATHOPHYSIOLOGICAL ROLE AND CLINICAL IMPLICATIONS [J].
BOHM, M .
KLINISCHE WOCHENSCHRIFT, 1987, 65 (11) :487-499
[10]  
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3