QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS BY DISTANCE GEOMETRY - SYSTEMATIC ANALYSIS OF DIHYDROFOLATE-REDUCTASE INHIBITORS

被引：41

作者：

CRIPPEN, GM

机构：

来源：

关键词：

D O I：

10.1021/jm00180a004

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：599 / 606

页数：8

共 7 条

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[3] DISTANCE GEOMETRY APPROACH TO RATIONALIZING BINDING DATA [J].

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HYNES, JB .

[5] QUINAZOLINES AS INHIBITORS OF DIHYDROFOLATE-REDUCTASE .2. [J].

HYNES, JB ;

ASHTON, WT ;

BRYANSMITH, D ;

FREISHEIM, JH .

[6]

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[7]

MARTIN YC, 1978, QUANTITATIVE DRUG DE