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EVIDENCE FOR THE METABOLIC-ACTIVATION OF NON-STEROIDAL ANTIOESTROGENS - A STUDY OF STRUCTURE-ACTIVITY-RELATIONSHIPS
被引:90
作者
:
ALLEN, KE
论文数:
0
引用数:
0
h-index:
0
ALLEN, KE
CLARK, ER
论文数:
0
引用数:
0
h-index:
0
CLARK, ER
JORDAN, VC
论文数:
0
引用数:
0
h-index:
0
JORDAN, VC
机构
:
来源
:
BRITISH JOURNAL OF PHARMACOLOGY
|
1980年
/ 71卷
/ 01期
关键词
:
D O I
:
10.1111/j.1476-5381.1980.tb10912.x
中图分类号
:
R9 [药学];
学科分类号
:
1007 ;
摘要
:
引用
收藏
页码:83 / 91
页数:9
相关论文
共 28 条
[1]
ADAM HK, 1979, BIOCHEM PHARMACOL, V27, P145
[2]
PREPARATION AND IDENTIFICATION OF CIS AND TRANS ISOMERS OF SUBSTITUTED TRIARYLETHYLENE
BEDFORD, GR
论文数:
0
引用数:
0
h-index:
0
BEDFORD, GR
RICHARDSON, DN
论文数:
0
引用数:
0
h-index:
0
RICHARDSON, DN
[J].
NATURE,
1966,
212
(5063)
: 733
-
+
[3]
CLOMIPHENE
BISHOP, PMF
论文数:
0
引用数:
0
h-index:
0
BISHOP, PMF
[J].
BRITISH MEDICAL BULLETIN,
1970,
26
(01)
: 22
-
&
[4]
INVESTIGATION OF AQUEOUS TWEEN 80 AS A VEHICLE FOR INTRAVAGINAL ADMINISTRATION
CLARK, ER
论文数:
0
引用数:
0
h-index:
0
CLARK, ER
MCCRACKEN, AM
论文数:
0
引用数:
0
h-index:
0
MCCRACKEN, AM
[J].
JOURNAL OF ENDOCRINOLOGY,
1971,
51
(04)
: 797
-
+
[5]
ANTIESTROGENIC AND ANTIFERTILITY COMPOUNDS .4. 1,1,2-TRIARYLALKAN-1-OLS AND 1,1,2-TRIARYLALK-1-ENES CONTAINING BASIC ETHER GROUPS
COLLINS, DJ
论文数:
0
引用数:
0
h-index:
0
COLLINS, DJ
HOBBS, JJ
论文数:
0
引用数:
0
h-index:
0
HOBBS, JJ
EMMENS, CW
论文数:
0
引用数:
0
h-index:
0
EMMENS, CW
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1971,
14
(10)
: 952
-
&
[6]
DIPACO G, 1962, Patent No. 9005903
[7]
UTEROTROPHIC ACTIVITY OF VARIOUS PHENOLIC STEROIDS
DORFMAN, RI
论文数:
0
引用数:
0
h-index:
0
DORFMAN, RI
KINCL, FA
论文数:
0
引用数:
0
h-index:
0
KINCL, FA
[J].
ACTA ENDOCRINOLOGICA,
1966,
52
(04):
: 619
-
&
[8]
ORAL-CONTRACEPTIVES - ETHINYL ESTRADIOL BINDS WITH HIGHER AFFINITY THAN MESTRANOL TO MACROMOLECULES FROM SITES OF ANTI-FERTILITY ACTION
EISENFELD, A
论文数:
0
引用数:
0
h-index:
0
机构:
YALE UNIV, SCH MED, DEPT PHARMACOL, NEW HAVEN, CT 06510 USA
YALE UNIV, SCH MED, DEPT PHARMACOL, NEW HAVEN, CT 06510 USA
EISENFELD, A
[J].
ENDOCRINOLOGY,
1974,
94
(03)
: 803
-
807
[9]
THE INTRAVAGINAL ASSAY OF NATURALLY OCCURRING OESTROGENS
EMMENS, CW
论文数:
0
引用数:
0
h-index:
0
EMMENS, CW
[J].
JOURNAL OF ENDOCRINOLOGY,
1950,
6
(03)
: 302
-
307
[10]
COMPARATIVE-STUDY OF ANTIESTROGEN ACTION - TEMPORAL PATTERNS OF ANTAGONISM OF ESTROGEN STIMULATED UTERINE GROWTH AND EFFECTS ON ESTROGEN-RECEPTOR LEVELS
FERGUSON, ER
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ILLINOIS, DEPT PHYSIOL & BIOPHYS, URBANA, IL 61801 USA
FERGUSON, ER
KATZENELLENBOGEN, BS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ILLINOIS, DEPT PHYSIOL & BIOPHYS, URBANA, IL 61801 USA
KATZENELLENBOGEN, BS
[J].
ENDOCRINOLOGY,
1977,
100
(05)
: 1242
-
1251
←
1
2
3
→
共 28 条
[1]
ADAM HK, 1979, BIOCHEM PHARMACOL, V27, P145
[2]
PREPARATION AND IDENTIFICATION OF CIS AND TRANS ISOMERS OF SUBSTITUTED TRIARYLETHYLENE
BEDFORD, GR
论文数:
0
引用数:
0
h-index:
0
BEDFORD, GR
RICHARDSON, DN
论文数:
0
引用数:
0
h-index:
0
RICHARDSON, DN
[J].
NATURE,
1966,
212
(5063)
: 733
-
+
[3]
CLOMIPHENE
BISHOP, PMF
论文数:
0
引用数:
0
h-index:
0
BISHOP, PMF
[J].
BRITISH MEDICAL BULLETIN,
1970,
26
(01)
: 22
-
&
[4]
INVESTIGATION OF AQUEOUS TWEEN 80 AS A VEHICLE FOR INTRAVAGINAL ADMINISTRATION
CLARK, ER
论文数:
0
引用数:
0
h-index:
0
CLARK, ER
MCCRACKEN, AM
论文数:
0
引用数:
0
h-index:
0
MCCRACKEN, AM
[J].
JOURNAL OF ENDOCRINOLOGY,
1971,
51
(04)
: 797
-
+
[5]
ANTIESTROGENIC AND ANTIFERTILITY COMPOUNDS .4. 1,1,2-TRIARYLALKAN-1-OLS AND 1,1,2-TRIARYLALK-1-ENES CONTAINING BASIC ETHER GROUPS
COLLINS, DJ
论文数:
0
引用数:
0
h-index:
0
COLLINS, DJ
HOBBS, JJ
论文数:
0
引用数:
0
h-index:
0
HOBBS, JJ
EMMENS, CW
论文数:
0
引用数:
0
h-index:
0
EMMENS, CW
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1971,
14
(10)
: 952
-
&
[6]
DIPACO G, 1962, Patent No. 9005903
[7]
UTEROTROPHIC ACTIVITY OF VARIOUS PHENOLIC STEROIDS
DORFMAN, RI
论文数:
0
引用数:
0
h-index:
0
DORFMAN, RI
KINCL, FA
论文数:
0
引用数:
0
h-index:
0
KINCL, FA
[J].
ACTA ENDOCRINOLOGICA,
1966,
52
(04):
: 619
-
&
[8]
ORAL-CONTRACEPTIVES - ETHINYL ESTRADIOL BINDS WITH HIGHER AFFINITY THAN MESTRANOL TO MACROMOLECULES FROM SITES OF ANTI-FERTILITY ACTION
EISENFELD, A
论文数:
0
引用数:
0
h-index:
0
机构:
YALE UNIV, SCH MED, DEPT PHARMACOL, NEW HAVEN, CT 06510 USA
YALE UNIV, SCH MED, DEPT PHARMACOL, NEW HAVEN, CT 06510 USA
EISENFELD, A
[J].
ENDOCRINOLOGY,
1974,
94
(03)
: 803
-
807
[9]
THE INTRAVAGINAL ASSAY OF NATURALLY OCCURRING OESTROGENS
EMMENS, CW
论文数:
0
引用数:
0
h-index:
0
EMMENS, CW
[J].
JOURNAL OF ENDOCRINOLOGY,
1950,
6
(03)
: 302
-
307
[10]
COMPARATIVE-STUDY OF ANTIESTROGEN ACTION - TEMPORAL PATTERNS OF ANTAGONISM OF ESTROGEN STIMULATED UTERINE GROWTH AND EFFECTS ON ESTROGEN-RECEPTOR LEVELS
FERGUSON, ER
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ILLINOIS, DEPT PHYSIOL & BIOPHYS, URBANA, IL 61801 USA
FERGUSON, ER
KATZENELLENBOGEN, BS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV ILLINOIS, DEPT PHYSIOL & BIOPHYS, URBANA, IL 61801 USA
KATZENELLENBOGEN, BS
[J].
ENDOCRINOLOGY,
1977,
100
(05)
: 1242
-
1251
←
1
2
3
→