ASSESSMENT OF MK-467, A PERIPHERAL ALPHA-2-ADRENOCEPTOR ANTAGONIST USING INTRAVENOUS CLONIDINE

被引:0
|
作者
WARREN, JB
DOLLERY, CT
SCIBERRAS, D
GOLDBERG, M
机构
[1] HAMMERSMITH HOSP,ROYAL POSTGRAD MED SCH,DEPT CLIN PHARMACOL,LONDON W12 0HS,ENGLAND
[2] HAMMERSMITH HOSP,ROYAL POSTGRAD MED SCH,DEPT MED,LONDON W12 0HS,ENGLAND
[3] MERCK SHARP & DOHME LTD,RAHWAY,NJ 07065
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:P306 / P306
页数:1
相关论文
共 50 条
  • [41] Effects of the peripherally acting α2-adrenoceptor antagonist MK-467 on cardiopulmonary function in sheep sedated by intramuscular administration of medetomidine and ketamine and reversed by intramuscular administration of atipamezole
    Adam, Magdy
    Raekallio, Marja R.
    Salla, Kati M.
    Honkavaara, Juhana M.
    Mannikko, Sofia
    Scheinin, Mika
    Kajula, Marena
    Molsa, Sari H.
    Vainio, Outi M.
    AMERICAN JOURNAL OF VETERINARY RESEARCH, 2018, 79 (09) : 921 - 932
  • [42] REVERSAL OF CLONIDINE-INDUCED EFFECTS IN HEALTHY-VOLUNTEERS BY RS-21361, A SELECTIVE ALPHA-2-ADRENOCEPTOR ANTAGONIST
    DOW, RJ
    WHITING, RL
    BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1984, 18 (02) : P288 - P288
  • [43] THE REVERSAL OF SOME CLONIDINE INDUCED EFFECTS BY SINGLE ORAL DOSES OF IDAZOXAN (RX781094), AN ALPHA-2-ADRENOCEPTOR ANTAGONIST
    CLIFFORD, JM
    PRICE, M
    BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1984, 17 (05) : P602 - P602
  • [44] BARORECEPTOR FUNCTION IN MAN FOLLOWING PERIPHERAL ALPHA-1-ADRENOCEPTOR AND ALPHA-2-ADRENOCEPTOR STIMULATION
    DEERING, AH
    RIDDELL, JG
    SHANKS, RG
    HARRON, DWG
    EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1987, 33 (01) : 41 - 47
  • [45] A PRELIMINARY, CLINICAL PHARMACOLOGICAL ASSESSMENT OF L-659,066, A NOVEL ALPHA-2-ADRENOCEPTOR ANTAGONIST
    SCHAFERS, RF
    ELLIOTT, HL
    HOWIE, CA
    REID, JL
    BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1992, 34 (06) : 521 - 526
  • [47] THE PHARMACOKINETICS AFTER INTRAVENOUS AND ORAL-ADMINISTRATION IN MAN OF THE ALPHA-2-ADRENOCEPTOR ANTAGONIST IDAZOXAN (RX781094)
    MUIR, NC
    LLOYDJONES, JG
    NICHOLS, JD
    CLIFFORD, JM
    EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1986, 29 (06) : 743 - 745
  • [48] STUDIES OF THE ALPHA-2-ADRENOCEPTOR AFFINITY AND THE ALPHA-2-ADRENOCEPTOR TO ALPHA-1-ADRENOCEPTOR SELECTIVITY OF SOME SUBSTITUTED BENZOQUINOLIZINES USING RECEPTOR-BINDING TECHNIQUES
    CHEUNG, YD
    NAHORSKI, SR
    RHODES, KF
    WATERFALL, JF
    BIOCHEMICAL PHARMACOLOGY, 1984, 33 (09) : 1566 - 1568
  • [49] REVERSAL OF SOME EFFECTS OF CLONIDINE BY RX781094, AN ALPHA-2-ADRENOCEPTOR ANTAGONIST - A PILOT-STUDY IN HEALTHY-VOLUNTEERS
    CLIFFORD, JM
    CROSSLEY, DI
    ORWIN, JM
    PRICE, M
    BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1982, 13 (04) : P609 - P609
  • [50] INFLUENCE OF ALPHA-1-ADRENOCEPTOR AND ALPHA-2-ADRENOCEPTOR ANTAGONIST THERAPY ON THE DEVELOPMENT OF HYPERTENSION IN SPONTANEOUSLY HYPERTENSIVE RATS
    YOUNG, RL
    JONSSON, JR
    MANO, MT
    FREWIN, DB
    HEAD, RJ
    JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1993, 21 (05) : 786 - 790