DEVELOPMENT OF TETRAZOLE BIOISOSTERES IN ANGIOTENSIN-II ANTAGONISTS

被引：17

作者：

FERRARI, B

TAILLADES, J

PERREAUT, P

BERNHART, C

GOUGAT, J

GUIRAUDOU, P

CAZAUBON, C

ROCCON, A

NISATO, D

LEFUR, G

BRELIERE, JC

机构：

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1994年 / 4卷 / 01期

关键词：

D O I：

10.1016/S0960-894X(01)81120-3

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

The application of acidic heterocycles as a substitute for tetrazole in the synthesis of potent non-peptide Angiotensin II AT1 receptor antagonists is described.

引用

页码：45 / 50

页数：6

共 15 条

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