TRICYCLIC QUINOXALINES AS LIGANDS FOR THE STRYCHNINE-INSENSITIVE GLYCINE SITE

被引：8

作者：

JACKSON, PF

DAVENPORT, TW

RESCH, JF

LEHR, GS

PULLAN, LM

机构：

[1] Biomedical Research Department, ICI Pharmaceuticals Group, Wilmington

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1991年 / 1卷 / 12期

关键词：

D O I：

10.1016/S0960-894X(01)81062-3

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

The synthesis of a series of tricyclic quinoxalines is described. These compounds exhibit good affinity for both the strychnine-insensitive glycine site of the NMDA receptor and the AMPA receptor.

引用

页码：751 / 756

页数：6

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