CONFORMATIONAL SHIFTS AT THE BENZODIAZEPINE RECEPTOR RELATED TO THE BINDING OF AGONISTS ANTAGONISTS AND INVERSE AGONISTS

被引：0
作者：
FRYER, RI
COOK, C
GILMAN, NW
WALSER, A
机构：
来源：
LIFE SCIENCES | 1986年 / 39卷 / 21期
关键词：
D O I：
暂无
中图分类号：
R-3 [医学研究方法]; R3 [基础医学];
学科分类号：
1001 ;
摘要：
引用
收藏
页码：1947 / 1957
页数：11
相关论文
共 50 条
[41]   Benzodiazepine receptor agonists and inverse agonists yield concordant rather than opposing effects on startle responses [J].
Berntson, G ;
Sarter, M ;
Ruland, S ;
Hart, S ;
Ronis, V .
JOURNAL OF PSYCHOPHARMACOLOGY, 1996, 10 (04) :309-312
[42]   The Neurochemical Mechanisms of the Pharmacological Activities of Inverse Agonists of the Benzodiazepine Binding Site [J].
Golovko, A. I. ;
Ivanov, M. B. ;
Golovko, E. S. ;
Dolgo-Saburov, V. B. ;
Zatsepin, E. P. .
NEUROCHEMICAL JOURNAL, 2018, 12 (04) :337-346
[43]   The Neurochemical Mechanisms of the Pharmacological Activities of Inverse Agonists of the Benzodiazepine Binding Site [J].
A. I. Golovko ;
M. B. Ivanov ;
E. S. Golovko ;
V. B. Dolgo-Saburov ;
E. P. Zatsepin .
Neurochemical Journal, 2018, 12 :337-346
[44]   SYNTHESIS OF 6-SUBSTITUTED BETA-CARBOLINES WHICH BEHAVE AS BENZODIAZEPINE RECEPTOR ANTAGONISTS OR INVERSE AGONISTS [J].
HAGEN, TJ ;
SKOLNICK, P ;
COOK, JM .
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1987, 193 :35-MEDI
[45]   THE EFFECT OF BENZODIAZEPINE AGONISTS AND INVERSE AGONISTS IN A RAT-FEEDING MODEL [J].
DEACON, RMJ ;
MCCULLOCH, AJ ;
GARDNER, CR .
PSYCHOPHARMACOLOGY, 1986, 89 (04) :S56-S56
[46]   BENZODIAZEPINE RECEPTORS - MODE OF INTERACTION OF AGONISTS AND ANTAGONISTS [J].
MOHLER, H .
ADVANCES IN BIOCHEMICAL PSYCHOPHARMACOLOGY, 1983, 37 :247-254
[47]   BIOMIMETIC APPROACH TO POTENTIAL BENZODIAZEPINE AGONISTS AND ANTAGONISTS [J].
CAIN, M ;
GUZMAN, F ;
COOK, JM ;
RICE, KC ;
SKOLNICK, P .
HETEROCYCLES, 1982, 19 (06) :1003-1007
[48]   Characterization of active and inactive states of CB1 receptor and the differential binding state modulation by cannabinoid agonists, antagonists and inverse agonists [J].
Gullapalli, Srinivas ;
Amrutkar, Dipak ;
Gupta, Sangeetha ;
Kandadi, Machender R. ;
Kumar, Hemant ;
Gandhi, Maulik ;
Karande, Vikas ;
Narayanan, Shridhar .
NEUROPHARMACOLOGY, 2010, 58 (08) :1215-1219
[49]   β3-ADRENOCEPTOR AGONISTS AND (ANTAGONISTS AS) INVERSE AGONISTS: HISTORY, PERSPECTIVE, CONSTITUTIVE ACTIVITY, AND STEREOSPECIFIC BINDING [J].
Perrone, Maria Grazia ;
Scilimati, Antonio .
METHODS IN ENZYMOLOGY, VOLUME 484: CONSTITUTIVE ACTIVITY IN RECEPTORS AND OTHER PROTEINS, PART A, 2010, 484 :197-230
[50]   DIFFERENTIAL MODULATION OF ETAZOLATE OR PENTOBARBITAL ENHANCED [H-3]MUSCIMOL BINDING BY BENZODIAZEPINE AGONISTS AND INVERSE AGONISTS [J].
BOREA, PA ;
SUPAVILAI, P ;
KAROBATH, M .
BRAIN RESEARCH, 1983, 280 (02) :383-386
12345