DESENSITIZATION OF PLATELETS TO ILOPROST - LOSS OF SPECIFIC BINDING-SITES AND HETEROLOGOUS DESENSITIZATION OF ADENYLATE-CYCLASE

被引:46
作者
JASCHONEK, K
FAUL, C
SCHMIDT, H
RENN, W
机构
关键词
D O I
10.1016/0014-2999(88)90777-7
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:187 / 196
页数:10
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共 36 条
[1]  
ALVAREZ R, 1981, MOL PHARMACOL, V20, P302
[2]  
BILLAH M M, 1979, Biochemical and Biophysical Research Communications, V90, P92, DOI 10.1016/0006-291X(79)91594-8
[3]  
BOEYNAEMS JM, 1980, OUTLINES RECEPTOR TH, P15
[4]  
CHAN SC, 1982, J CYCLIC NUCL PROT, V8, P211
[5]  
CLARK RB, 1979, J BIOL CHEM, V254, P9373
[6]  
DARFLER FJ, 1982, J BIOL CHEM, V257, P1901
[7]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[8]   PROSTACYCLIN ANALOGS REDUCE ADP-RIBOSYLATION OF THE ALPHA-SUBUNIT OF THE REGULATORY GS-PROTEIN AND DIMINISH ADENOSINE (A2) RESPONSIVENESS OF PLATELETS [J].
EDWARDS, RJ ;
MACDERMOT, J ;
WILKINS, AJ .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 90 (03) :501-510
[9]   THE CYTOPLASMIC CONCENTRATION OF FREE CALCIUM IN PLATELETS IS CONTROLLED BY STIMULATORS OF CYCLIC-AMP PRODUCTION (PGD2, PGE1, FORSKOLIN) [J].
FEINSTEIN, MB ;
EGAN, JJ ;
SHAAFI, RI ;
WHITE, J .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1983, 113 (02) :598-604
[10]  
GARRITY M, 1983, J BIOL CHEM, V258, P8692