AF-DX 116 DISCRIMINATES BETWEEN MUSCARINIC M2-RECEPTORS OF THE HEART AND VASCULATURE

被引:40
作者
DUCKLES, SP [1 ]
YAMAMURA, HI [1 ]
LEE, V [1 ]
机构
[1] UNIV ARIZONA,COLL MED,DEPT PHARMACOL,TUCSON,AZ 85724
关键词
D O I
10.1016/0024-3205(87)90383-3
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:1507 / 1511
页数:5
相关论文
共 13 条
[1]   VASODILATATION BY ACETYLCHOLINE IS ENDOTHELIUM-DEPENDENT - A STUDY BY SONOMICROMETRY IN CANINE FEMORAL-ARTERY INVIVO [J].
ANGUS, JA ;
CAMPBELL, GR ;
COCKS, TM ;
MANDERSON, JA .
JOURNAL OF PHYSIOLOGY-LONDON, 1983, 344 (NOV) :209-&
[2]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[3]  
EGLEN RM, 1984, BR J PHARM, V71, P141
[5]   THE OBLIGATORY ROLE OF ENDOTHELIAL-CELLS IN THE RELAXATION OF ARTERIAL SMOOTH-MUSCLE BY ACETYLCHOLINE [J].
FURCHGOTT, RF ;
ZAWADZKI, JV .
NATURE, 1980, 288 (5789) :373-376
[6]  
FURCHGOTT RF, 1972, CATECHOLAMINES, P283
[7]   CARDIOSELECTIVE PROFILE OF AF-DX-116, A MUSCARINE M2 RECEPTOR ANTAGONIST [J].
GIACHETTI, A ;
MICHELETTI, R ;
MONTAGNA, E .
LIFE SCIENCES, 1986, 38 (18) :1663-1672
[8]   MUSCARINIC RECEPTOR SUBTYPES - M1 AND M2 BIOCHEMICAL AND FUNCTIONAL-CHARACTERIZATION [J].
HAMMER, R ;
GIACHETTI, A .
LIFE SCIENCES, 1982, 31 (26) :2991-2998
[9]   PIRENZEPINE DISTINGUISHES BETWEEN DIFFERENT SUBCLASSES OF MUSCARINIC RECEPTORS [J].
HAMMER, R ;
BERRIE, CP ;
BIRDSALL, NJM ;
BURGEN, ASV ;
HULME, EC .
NATURE, 1980, 283 (5742) :90-92
[10]  
HYNES MR, 1986, J PHARMACOL EXP THER, V238, P100