CHIRAL SYNTHESIS OF D-3,3-DIPHENYLALANINE AND L-3,3-DIPHENYLALANINE (DIP), UNUSUAL ALPHA-AMINO-ACIDS FOR PEPTIDES OF BIOLOGICAL INTEREST

被引：37

作者：

CHEN, HG ^{[1
]}

BEYLIN, VG ^{[1
]}

MARLATT, M ^{[1
]}

LEJA, B ^{[1
]}

GOEL, OP ^{[1
]}

机构：

[1] WARNER LAMBERT PARKE DAVIS, PARKE DAVIS PHARMACEUT RES DIV, 2800 PLYMOUTH RD, ANN ARBOR, MI 48105 USA

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 23期

关键词：

D O I：

10.1016/S0040-4039(00)92070-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The asymmetric syntheses of D-(R)-(-)- and L-(S)-(+)-3,3-diphenylalanine (Dip)

引用

页码：3293 / 3296

页数：4

共 10 条

[1]

CZARNIECKI MF, 1989, Patent No. 4766109

[2] THE TOTAL SYNTHESES OF THE ISODITYROSINE-DERIVED CYCLIC TRIPEPTIDES OF4949-III AND K-13 - DETERMINATION OF THE ABSOLUTE-CONFIGURATION OF K-13 [J].

EVANS, DA ;

ELLMAN, JA .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1989, 111 (03) :1063-1072

[3] THE ASYMMETRIC-SYNTHESIS OF ALPHA-AMINO-ACIDS - ELECTROPHILIC AZIDATION OF CHIRAL IMIDE ENOLATES, A PRACTICAL APPROACH TO THE SYNTHESIS OF (R)-ALPHA-AZIDO AND (S)-ALPHA-AZIDO CARBOXYLIC-ACIDS [J].

EVANS, DA ;

BRITTON, TC ;

ELLMAN, JA ;

DOROW, RL .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1990, 112 (10) :4011-4030

[4] EVALUATION OF A CHIRAL CROWN-ETHER LC COLUMN FOR THE SEPARATION OF RACEMIC AMINES [J].

HILTON, M ;

ARMSTRONG, DW .

JOURNAL OF LIQUID CHROMATOGRAPHY, 1991, 14 (01) :9-28

[5] EMERGING APPROACHES IN THE MOLECULAR DESIGN OF RECEPTOR-SELECTIVE PEPTIDE LIGANDS - CONFORMATIONAL, TOPOGRAPHICAL AND DYNAMIC CONSIDERATIONS [J].

HRUBY, VJ ;

ALOBEIDI, F ;

KAZMIERSKI, W .

BIOCHEMICAL JOURNAL, 1990, 268 (02) :249-262

[6] TOPOGRAPHIC PROBES OF ANGIOTENSIN AND RECEPTOR - POTENT ANGIOTENSIN-II AGONIST CONTAINING DIPHENYLALANINE AND LONG-ACTING ANTAGONISTS CONTAINING BIPHENYLALANINE AND 2-INDAN AMINO-ACID IN POSITION 8 [J].

HSIEH, KH ;

LAHANN, TR ;

SPETH, RC .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (04) :898-903

[7] ASYMMETRIC-SYNTHESIS OF L-DIPHENYLALANINE AND L-9-FLUORENYLGLYCINE VIA ROOM-TEMPERATURE ALKYLATIONS OF A SULTAM-DERIVED GLYCINE IMINE [J].

JOSIEN, H ;

MARTIN, A ;

CHASSAING, G .

TETRAHEDRON LETTERS, 1991, 32 (45) :6547-6550

[8] ASYMMETRIC-SYNTHESIS OF TOPOGRAPHICALLY CONSTRAINED AMINO-ACIDS - SYNTHESIS OF THE OPTICALLY PURE ISOMERS OF ALPHA,BETA-DIMETHYL-PHENYLALANINE AND ALPHA,BETA-DIMETHYL-1,2,3,4-TETRAHYDROISOQUINOLINE-3-CARBOXYLIC ACID [J].

KAZMIERSKI, WM ;

HRUBY, VJ .

TETRAHEDRON LETTERS, 1991, 32 (41) :5769-5772

[9] CHROMATOGRAPHIC-SEPARATION OF RACEMIC AMINO-ACIDS BY USE OF CHIRAL CROWN ETHER-COATED REVERSED-PHASE PACKINGS [J].

SHINBO, T ;

YAMAGUCHI, T ;

NISHIMURA, K ;

SUGIURA, M .

JOURNAL OF CHROMATOGRAPHY, 1987, 405 :145-153

[10]

003 DAIC CHEM IND LT

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