8-PIPERAZINYL-2,3-DIHYDRO-1,4-DIOXINO[2,3-B]PYRIDINE DERIVATIVES - SYNTHESIS AND INTERACTION WITH 5-HT SEROTONIN BINDING-SITES

被引:0
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作者
JOSEPH, B
BENARAB, A
GUILLAUMET, G
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O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The synthesis of 8-piperazinyl-2,3-dihydro-1,4-dioxino[2,3-b]pyridine derivatives (6a-c) are described. Their affinity and selectivity for 5-HT serotoninergic sites were evaluated.
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页码:1355 / 1360
页数:6
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