SYNTHESIS OF A NOVEL SERIES OF TOPOGRAPHICALLY CONSTRAINED AMINO-ACIDS - BENZO-1,2,3,4-TETRAHYDROISOQUINOLINE-3-CARBOXYLIC ACIDS

被引：0

作者：

WANG, CG ^{[1
]}

MOSBERG, HI ^{[1
]}

机构：

[1] UNIV MICHIGAN,COLL PHARM,ANN ARBOR,MI 48105

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 21期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A novel series of benzo-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids (benzo Tic, Figure 1), designed by extending the aromatic system of Tic (Tic = 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid) in three different orientations, has been synthesized.

引用

页码：3623 / 3626

页数：4

共 9 条

[1] SYNTHESIS OF PHENYLALANINE ANALOGS AS ANTIMETABOLITES
BURCKHALTER, JH
STEPHENS, VC
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1951, 73 (01) : 56 - 58
[2] SIDE-CHAIN BROMINATION OF SOME ALKYLNAPHTHALENES WITH N-BROMOSUCCINIMIDE
BUUHOI, NP
LECOCQ, J
[J]. JOURNAL OF THE CHEMICAL SOCIETY, 1946, (SEP): : 830 - 832
[3] A NEW APPROACH TO RECEPTOR LIGAND DESIGN - SYNTHESIS AND CONFORMATION OF A NEW CLASS OF POTENT AND HIGHLY SELECTIVE MU-OPIOID ANTAGONISTS UTILIZING TETRAHYDROISOQUINOLINE CARBOXYLIC-ACID
KAZMIERSKI, W
HRUBY, VJ
[J]. TETRAHEDRON, 1988, 44 (03) : 697 - 710
[4] PROBING THE BRADYKININ RECEPTOR - MAPPING THE GEOMETRIC TOPOGRAPHY USING ETHERS OF HYDROXYPROLINE IN NOVEL PEPTIDES
KYLE, DJ
MARTIN, JA
BURCH, RM
CARTER, JP
LU, SF
MEEKER, S
PROSSER, JC
SULLIVAN, JP
TOGO, J
NORONHABLOB, L
SINSKO, JA
WALTERS, RF
WHALEY, LW
HINER, RN
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1991, 34 (08) : 2649 - 2653
[5] MOSBERG HI, 1994, LETT PEPT SCI, V1, P67
[6] Studies in the phenanthrene series XXII Derivatives of dibenzisoquinoline and naphthisoquinoline
Mosettig, E
May, EL
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1938, 60 : 2962 - 2966
[7] On the formation of isochinolin-derivatives through the development of methylial on phenyl-aether, phenyl-alanin and tyrosin.
Pictet, A
Spengler, T
[J]. BERICHTE DER DEUTSCHEN CHEMISCHEN GESELLSCHAFT, 1911, 44 : 2030 - 2036
[8] SCHILLER PW, 1992, PEPTIDE CHEM, P337
[9] CONVERSION OF ENKEPHALIN AND DERMORPHIN INTO DELTA-SELECTIVE OPIOID ANTAGONISTS BY SINGLE-RESIDUE SUBSTITUTION
TANCREDI, T
SALVADORI, S
AMODEO, P
PICONE, D
LAZARUS, LH
BRYANT, SD
GUERRINI, R
MARZOLA, G
TEMUSSI, PA
[J]. EUROPEAN JOURNAL OF BIOCHEMISTRY, 1994, 224 (01): : 241 - 247

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