STEREOCHEMICAL STUDIES ON MEDICINAL AGENTS .17. SYNTHESIS, ABSOLUTE-CONFIGURATION, AND ANALGETIC POTENCY OF ENANTIOMERIC DIASTEREOMERS OF 3-ETHYL AND 3-PROPYL DERIVATIVES OF 1-METHYL-4-PHENYL-4-PROPIONOXYPIPERIDINE

被引：15

作者：

BELL, KH ^{[1
]}

PORTOGHESE, PS ^{[1
]}

机构：

[1] UNIV MINNESOTA, COLL PHARM, DEPT MED CHEM, MINNEAPOLIS, MN 55455 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1974年 / 17卷 / 01期

关键词：

D O I：

10.1021/jm00247a024

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：129 / 131

页数：3

共 8 条

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[2] STEREOCHEMICAL STUDIES ON MEDICINAL AGENTS .15. ABSOLUTE-CONFIGURATIONS AND ANALGETIC POTENCIES OF ENANTIOMERIC DIASTEREOMERS OF 3-ALLYL-1-METHYL-4-PHENYL-4-PROPIONOXYPIPERIDINE [J].

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[6] STEREOCHEMICAL STUDIES ON MEDICINAL AGENTS .12. DISTINCTION OF ENANTIOTOPIC GROUPS IN INTERACTION OF 1-METHYL-4-PHENYL-4-PROPIONOXYPIPERIDINE WITH ANALGETIC RECEPTORS [J].

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[7] STEREOCHEMICAL STUDIES ON MEDICINAL AGENTS .13. CORRELATION OF SOLID-STATE CONFORMATIONS OF 1,3,5-TRIMETHYL-4-PHENYL-4-PROPIONOXYPIPERIDINE AND 1,3-DIMETHYL-4-PHENYL-4-PROPIONOXYPIPERIDINE ENANTIOMERS WITH THEIR ABSOLUTE STEREOSELECTIVITY AT ANALGETIC RECEPTORS [J].

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[8] PIPERIDINE DERIVATIVES .4. 1,3-DISUBSTITUTED-4-ARYL-4-ACYLOXY PIPERIDINES [J].

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