TISSUE SELECTIVITY OF THE CHOLESTEROL-LOWERING AGENTS LOVASTATIN, SIMVASTATIN AND PRAVASTATIN IN RATS INVIVO

被引:158
作者
GERMERSHAUSEN, JI
HUNT, VM
BOSTEDOR, RG
BAILEY, PJ
KARKAS, JD
ALBERTS, AW
机构
关键词
D O I
10.1016/0006-291X(89)92773-3
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:667 / 675
页数:9
相关论文
共 12 条
[1]   MEVINOLIN - A HIGHLY POTENT COMPETITIVE INHIBITOR OF HYDROXYMETHYLGLUTARYL-COENZYME-A REDUCTASE AND A CHOLESTEROL-LOWERING AGENT [J].
ALBERTS, AW ;
CHEN, J ;
KURON, G ;
HUNT, V ;
HUFF, J ;
HOFFMAN, C ;
ROTHROCK, J ;
LOPEZ, M ;
JOSHUA, H ;
HARRIS, E ;
PATCHETT, A ;
MONAGHAN, R ;
CURRIE, S ;
STAPLEY, E ;
ALBERSSCHONBERG, G ;
HENSENS, O ;
HIRSHFIELD, J ;
HOOGSTEEN, K ;
LIESCH, J ;
SPRINGER, J .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (07) :3957-3961
[2]  
BROWN AG, 1976, J CHEM SOC PERK T, V1, P1165
[3]   MONACOLIN-K, A NEW HYPOCHOLESTEROLEMIC AGENT PRODUCED BY A MONASCUS SPECIES [J].
ENDO, A .
JOURNAL OF ANTIBIOTICS, 1979, 32 (08) :852-854
[4]   ML-236A, ML-236B, AND ML-236C, NEW INHIBITORS OF CHOLESTEROGENESIS PRODUCED BY PENICILLIUM CITRINUM [J].
ENDO, A ;
KURODA, M ;
TSUJITA, Y .
JOURNAL OF ANTIBIOTICS, 1976, 29 (12) :1346-1348
[5]  
HARUYAMA H, 1986, CHEM PHARM BULL, V34, P1459
[6]  
HELLER RA, 1976, J BIOL CHEM, V251, P3815
[7]  
HOFFMAN WF, 1986, J MED CHEM, V29, P849, DOI 10.1021/jm00155a040
[8]   PURIFICATION OF 3-HYDROXY-3-METHYLGLUTARYL-COENZYME-A REDUCTASE FROM RAT-LIVER [J].
KLEINSEK, DA ;
RANGANATHAN, S ;
PORTER, JW .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (04) :1431-1435
[9]   MICROBIAL HYDROXYLATION OF ML-236B (COMPACTIN) - STUDIES ON MICROORGANISMS CAPABLE OF 3-BETA-HYDROXYLATION OF ML-236B [J].
SERIZAWA, N ;
SERIZAWA, S ;
NAKAGAWA, K ;
FURUYA, K ;
OKAZAKI, T ;
TERAHARA, A .
JOURNAL OF ANTIBIOTICS, 1983, 36 (07) :887-891