MOLECULAR MECHANISM OF INHIBITION OF RNASE-H ACTIVITY OF HIV-1 REVERSE-TRANSCRIPTASE BY AZTMP

被引:0
作者
ZHAN, XY [1 ]
TAN, CK [1 ]
DOWNEY, KM [1 ]
SO, AG [1 ]
机构
[1] UNIV MIAMI,DEPT MED R99,MIAMI,FL 33136
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:178 / 178
页数:1
相关论文
共 50 条
[31]   ILLIMAQUINONE, A SELECTIVE INHIBITOR OF THE RNASE-H ACTIVITY OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REVERSE-TRANSCRIPTASE [J].
LOYA, S ;
TAL, R ;
KASHMAN, Y ;
HIZI, A .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1990, 34 (10) :2009-2012
[32]   FIDELITY OF HIV-1 REVERSE-TRANSCRIPTASE [J].
PRESTON, BD ;
POIESZ, BJ ;
LOEB, LA .
SCIENCE, 1988, 242 (4882) :1168-1171
[33]   DETERMINANTS OF THE RNASE-H CLEAVAGE SPECIFICITY OF HUMAN-IMMUNODEFICIENCY-VIRUS REVERSE-TRANSCRIPTASE [J].
DESTEFANO, JJ ;
MALLABER, LM ;
FAY, PJ ;
BAMBARA, RA .
NUCLEIC ACIDS RESEARCH, 1993, 21 (18) :4330-4338
[34]   HIV-1 REVERSE TRANSCRIPTASE-ASSOCIATED RNASE-H CLEAVES RNA/RNA IN ARRESTED COMPLEXES - IMPLICATIONS FOR THE MECHANISM BY WHICH RNASE-H DISCRIMINATES BEWEEN RNA/RNA AND RNA/DNA [J].
GOTTE, M ;
FACKLER, S ;
HERMANN, T ;
PEROLA, E ;
CELLAI, L ;
GROSS, HJ ;
LEGRICE, SFJ ;
HEUMANN, H .
EMBO JOURNAL, 1995, 14 (04) :833-841
[35]   PHOSPHOROTHIOATE ANALOGS OF 2-5A - ACTIVATION INHIBITION OF RNASE-L AND INHIBITION OF HIV-1 REVERSE-TRANSCRIPTASE [J].
SUHADOLNIK, RJ ;
LEBLEU, B ;
PFLEIDERER, W ;
CHARUBALA, R ;
MONTEFIORI, DC ;
MITCHELL, WM ;
SOBOL, RW ;
LI, SW ;
KARIKO, K ;
REICHENBACH, NL .
NUCLEOSIDES & NUCLEOTIDES, 1989, 8 (5-6) :987-990
[36]   STRUCTURE OF THE RIBONUCLEASE H DOMAIN OF HIV-1 REVERSE-TRANSCRIPTASE [J].
MATTHEWS, DA ;
HOSTOMSKA, Z ;
HOSTOMSKY, Z ;
DAVIES, J ;
JORDAN, S .
FASEB JOURNAL, 1992, 6 (01) :A266-A266
[37]   SYNTHESIS AND HIV-1 REVERSE-TRANSCRIPTASE INHIBITION-ACTIVITY OF FUNCTIONALIZED PYROPHOSPHATE ANALOGS [J].
MCKENNA, CE ;
KHARE, A ;
JU, JY ;
LI, ZM ;
DUNCAN, G ;
CHENG, YC ;
KILKUSKIE, R .
PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS, 1993, 76 (1-4) :399-402
[38]   Inhibitory effects of quinones on RNase H activity associated with HIV-1 reverse transcriptase [J].
Min, BS ;
Miyashiro, H ;
Hattori, M .
PHYTOTHERAPY RESEARCH, 2002, 16 :S57-S62
[39]   STRUCTURE-ACTIVITY ANALYSES OF HIV-1 REVERSE-TRANSCRIPTASE [J].
BASU, A ;
BASU, S ;
MODAK, MJ .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1992, 183 (03) :1131-1138
[40]   PHOSPHOROTHIOATE OLIGONUCLEOTIDES BLOCK REVERSE TRANSCRIPTION BY THE RNASE-H ACTIVITY ASSOCIATED WITH THE HIV-1 POLYMERASE [J].
HATTA, T ;
TAKAI, K ;
YOKOYAMA, S ;
NAKASHIMA, H ;
YAMAMOTO, N ;
TAKAKU, H .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1995, 211 (03) :1041-1046