THE ASYMMETRIC-SYNTHESIS OF NONPEPTIDE CCK-A RECEPTOR AGONISTS

被引:11
作者
BURGAUD, BGM
HORWELL, DC
PRITCHARD, MC
BERNAD, N
MARTINEZ, J
机构
[1] ADDENBROOKES HOSP,PARKE DAVIS NEUROSCI RES CTR,CAMBRIDGE CB2 2QB,ENGLAND
[2] FAC PHARM MONTPELLIER,CNRS,URA,F-34060 MONTPELLIER,FRANCE
关键词
D O I
10.1016/0957-4166(95)00130-H
中图分类号
O61 [无机化学];
学科分类号
070301 ; 081704 ;
摘要
The asymmetric synthesis, CCK receptor binding affinities and CCK-A agonist properties of a novel series of non-peptide CCK-A receptor selective ligands is reported.
引用
收藏
页码:1081 / 1084
页数:4
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