ANTAGONISM OF ESTROGEN-RECEPTOR BINDING TO DNA AND ESTROGEN RESPONSE ELEMENT-DEPENDENT TRANSCRIPTION BY A NOVEL SUBSTITUTED INDOLE IS UNRELATED TO BINDING OF ESTRADIOL TO ITS RECEPTOR

被引:0
|
作者
BITONTI, AJ [1 ]
DUMONT, JA [1 ]
SALITURO, FG [1 ]
MCDONALD, IA [1 ]
WRIGHT, PS [1 ]
BAUMANN, RJ [1 ]
机构
[1] MARION MERRELL DOW RES INST,CINCINNATI,OH 45215
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:235 / 235
页数:1
相关论文
共 50 条
  • [1] ESTROGEN-RECEPTOR BINDING TO A DNA RESPONSE ELEMENT INVITRO IS NOT DEPENDENT UPON ESTRADIOL
    MURDOCH, FE
    MEIER, DA
    FURLOW, JD
    GRUNWALD, KAA
    GORSKI, J
    BIOCHEMISTRY, 1990, 29 (36) : 8377 - 8385
  • [2] MODULATION OF ESTROGEN-RECEPTOR BINDING TO DNA BY ESTRADIOL
    SKAFAR, DF
    NOTIDES, AC
    FEDERATION PROCEEDINGS, 1985, 44 (05) : 1473 - 1473
  • [3] SPECIFIC BINDING OF ESTROGEN-RECEPTOR TO THE ESTROGEN RESPONSE ELEMENT
    KLEINHITPASS, L
    TSAI, SY
    GREENE, GL
    CLARK, JH
    TSAI, MJ
    OMALLEY, BW
    MOLECULAR AND CELLULAR BIOLOGY, 1989, 9 (01) : 43 - 49
  • [4] BINDING OF THE ESTROGEN-RECEPTOR DNA-BINDING DOMAIN TO THE ESTROGEN RESPONSE ELEMENT INDUCES DNA BENDING
    NARDULLI, AM
    SHAPIRO, DJ
    MOLECULAR AND CELLULAR BIOLOGY, 1992, 12 (05) : 2037 - 2042
  • [5] Prebending the estrogen response element destabilizes binding of the estrogen receptor DNA binding domain
    Kim, J
    deHaan, G
    Nardulli, AM
    Shapiro, DJ
    MOLECULAR AND CELLULAR BIOLOGY, 1997, 17 (06) : 3173 - 3180
  • [6] THE ALLOSTERIC ESTROGEN-BINDING AND DNA-BINDING MECHANISM OF THE ESTROGEN-RECEPTOR
    SKAFAR, DF
    NOTIDES, AC
    BIOCHEMICAL ACTIONS OF HORMONES, 1987, 14 : 317 - 348
  • [7] BINDING OF ESTRADIOL-PEROXIDASE CONJUGATE TO ESTROGEN-RECEPTOR
    BHATTACHARJEE, M
    ALI, E
    JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1990, 37 (05): : 693 - 696
  • [8] BIOCHEMICAL SIMILARITIES OF ESTRADIOL BINDING TO ESTROGEN-RECEPTOR AND TYROSINASE
    ZAVA, DT
    GOLDHIRSCH, A
    PROCEEDINGS OF THE AMERICAN ASSOCIATION FOR CANCER RESEARCH, 1983, 24 (MAR): : 181 - 181
  • [9] CYANOKETONE COMPETITION WITH ESTRADIOL FOR BINDING TO THE CYTOSOLIC ESTROGEN-RECEPTOR
    WOLFSON, AJ
    RICHARDS, J
    ROTENSTEIN, D
    JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1983, 19 (06): : 1817 - 1818
  • [10] Binding of estrogen receptor β to estrogen response element in situ is independent of estradiol and impaired by its amino terminus
    Huang, J
    Li, XD
    Maguire, CA
    Hilf, R
    Bambara, RA
    Muyan, M
    MOLECULAR ENDOCRINOLOGY, 2005, 19 (11) : 2696 - 2712