(S)-5-PYRROLIDIN-2-YL-1H-TETRAZOLE

被引：18

作者：

Aureggi, Valentina ^{[2
]}

Franckevicius, Vilius ^{[3
]}

Kitching, Matthew O.

Ley, Steven V. ^{[1
]}

Longbottom, Deborah A. ^{[4
]}

Oelke, Alexander J. ^{[5
]}

Sedelmeier, Gottfried ^{[6
]}

机构：

[1] Univ Cambridge, Trinity Coll, Cambridge, England

[2] Univ Toronto, Prof Mark Lautenss Grp, Toronto, ON, Canada

[3] Ley Grp, Applicat Organocatalyt Methodol Nat Prod Synth, Cambridge, England

[4] Homerton Coll, Dept Chem, Cambridge, England

[5] Univ Cambridge, Applicat Organocatalyt Methodol Nat Prod Synth, Cambridge, England

[6] Univ Freiburg, Breisgau, Germany

来源：

ORGANIC SYNTHESES | 2008年 / 85卷

关键词：

D O I：

10.15227/orgsyn.085.0072

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：72 / +

页数：31

共 35 条

[1] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CARBOXYLIC-ACID REPLACEMENT ANALOGS OF THE POTENT ANGIOTENSIN CONVERTING ENZYME-INHIBITOR 5(S)-BENZAMIDO-4-OXO-6-PHENYLHEXANOYL-L-PROLINE [J].

ALMQUIST, RG ;

CHAO, WR ;

JENNINGSWHITE, C .

JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (08) :1067-1071

[2]

[Anonymous], PROC R D CHEM AN DEV

[3] The process development of RG 12525 (2-{[4-(tetrazol-5-ylmethylphenyl)-methoxy]phenoxymethyl}quinoline) [J].

Bridge, AW ;

Jones, RH ;

Kabir, H ;

Kee, AA ;

Lythgoe, DJ ;

Nakach, M ;

Pemberton, C ;

Wrightman, JA .

ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2001, 5 (01) :9-15

[4] Total synthesis of LFA-1 antagonist BIRT-377 via organocatalytic asymmetric construction of a quaternary stereocenter [J].

Chowdari, NS ;

Barbas, CF .

ORGANIC LETTERS, 2005, 7 (05) :867-870

[5] Organocatalysis with proline derivatives: improved catalysts for the asymmetric Mannich, nitro-Michael and aldol reactions [J].

Cobb, AJA ;

Shaw, DM ;

Longbottom, DA ;

Gold, JB ;

Ley, SV .

ORGANIC & BIOMOLECULAR CHEMISTRY, 2005, 3 (01) :84-96

[6] 5-Pyrrolidin-2-yltetrazole as an asymmetric organocatalyst for the addition of ketones to nitro-olefins [J].

Cobb, AJA ;

Longbottom, DA ;

Shaw, DM ;

Ley, SV .

CHEMICAL COMMUNICATIONS, 2004, (16) :1808-1809

[7] 5-pyrrolidin-2-yltetrazole: A new, catalytic, more soluble alternative to proline in an organocatalytic asymmetric Mannich-type reaction [J].

Cobb, AJA ;

Shaw, DM ;

Ley, SV .

SYNLETT, 2004, (03) :558-560

[8] An expedient route to the tetrazole analogues of α-amino acids [J].

Demko, ZP ;

Sharpless, KB .

ORGANIC LETTERS, 2002, 4 (15) :2525-2527

[9] Practical synthesis of (S)-pyrrolidin-2-yl-1H-tetrazole, incorporating efficient protecting group removal by flow-reactor hydrogenolysis [J].

Franckevicius, V ;

Knudsen, KR ;

Ladlow, M ;

Longbottom, DA ;

Ley, SV .

SYNLETT, 2006, (06) :889-892

[10]

GRZONKA Z, 1978, POL J CHEM, V52, P1412

← 1 2 3 4 →