THE SYNTHESIS OF 1-(3,4-DIHYDROXYPHENYL)-2-PROPANONE AND 1-(3,4-DIHYDROXYPHENYL)-2-PROPANOL

被引：0
|
作者：
BROZDA, D
机构：
来源：
PHARMAZIE | 1994年 / 49卷 / 08期
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中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
Acetylation of 1,3-propylenedithioacetal of 3,4-dihydroxybenzaldehyde silyl ether 5 followed by reductive desulfurization of the masking group gave ketone 7 which was reduced to alcohol 8. Hydrolysis of the silyl protecting groups in 7 and 8 afforded the title compounds which wer metabolites of 1-(4-hydroxy-3-methoxyphenyl)-2-propanone, found in smoked meat.
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页码：573 / 575
页数：3
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