SYNTHESIS OF NEW HETEROCYCLIC SCHIFF BASE, THIAZOLIDINONE AND AZETIDINONE COMPOUNDS AND THEIR ANTIBACTERIAL ACTIVITY AND ANTI-HIV ACTIVITIES

被引：0
|
作者：
Patel, Rajarshi N. [1 ]
Patel, P. V. [2 ]
Desai, K. R. [2 ]
Purohit, P. Y. [2 ]
Nimavat, K. S. [3 ]
Vyas, K. B. [4 ]
机构：
[1] Suleshvari Pharm, Ankleshwar 393002, Gujarat, India
[2] South Gujarat Univ, Dept Chem, Surat 395007, India
[3] Govt Sci Coll, Dept Chem, Gandhinagar 382015, Gujarat, India
[4] Sheth LH Sci Collage, Dept Chem, Mansa 382845, Gujarat, India
来源：
HETEROCYCLIC LETTERS | 2012年 / 2卷 / 01期
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中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Thiazolidines and azetidinopnes have been prepared by the reaction of various Schiff bases with thioglycine acid chloroacetyl chloride respectively. The intermediate Schiff bases were synthesized by the condensation of 4-amino-2,4'-dichloro diphenyl ether with various aldehydes. The structures of the compounds have been confirmed by elemental analysis and spectral analysis. The antibacterial and anti HIV activities of the compounds have been also screened.
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页码：99 / 105
页数：7
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