FLUORINATED PYRIMIDINES AS TIGHT-BINDING INHIBITORS OF THYMIDYLATE SYNTHETASE

被引：67

作者：

DANENBERG, PV ^{[1
]}

LOCKSHIN, A ^{[1
]}

机构：

[1] UNIV SO CALIF,SCH MED,CTR COMPREHENS CANC,LOS ANGELES,CA 90033

来源：

PHARMACOLOGY & THERAPEUTICS | 1981年 / 13卷 / 01期

关键词：

D O I：

10.1016/0163-7258(81)90068-1

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

收藏

页码：69 / 90

页数：22

相关论文

共 89 条

[1] SUICIDE ENZYME INACTIVATORS
ABELES, RH
MAYCOCK, AL
[J]. ACCOUNTS OF CHEMICAL RESEARCH, 1976, 9 (09) : 313 - 319
[2] ACKERMANN WW, 1949, P SOC EXP BIOL MED, V72, P1
[3] ALDRIDGE WN, 1972, FRONT BIOL, V26, P91
[4] THE SYNTHESIS OF NUCLEOSIDE AND NUCLEOTIDE ANALOGS DERIVED FROM URIDINE
BANNISTER, B
KAGAN, F
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1960, 82 (13) : 3363 - 3368
[5] CALORIMETRIC STUDY OF BINDING OF 2'-DEOXYURIDINE-5'-PHOSPHATE AND 5-FLUORO-2'-DEOXYURIDINE-5'-PHOSPHATE TO THYMIDYLATE SYNTHETASE
BEAUDETTE, NV
LANGERMAN, N
KISLIUK, RL
GAUMONT, Y
[J]. ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1977, 179 (01) : 272 - 278
[6] BELLISARIO RL, 1979, J BIOL CHEM, V254, P1296
[7] AMINO-ACID SEQUENCE AT FDUMP BINDING-SITE OF THYMIDYLATE SYNTHETASE
BELLISARIO, RL
MALEY, GF
GALIVAN, JH
MALEY, F
[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1976, 73 (06) : 1848 - 1852
[8] BLAKLEY RL, 1963, J BIOL CHEM, V238, P2113
[9] BRUICE TW, 1978, 6TH INT S CHEM BIOL
[10] ELUCIDATION OF DETAILED STRUCTURES OF NATIVE AND DENATURED TERNARY COMPLEXES OF THYMIDYLATE SYNTHETASE VIA F-19 NMR
BYRD, RA
DAWSON, WH
ELLIS, PD
DUNLAP, RB
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1978, 100 (24) : 7478 - 7486

← 1 2 3 4 5 6 7 8 9 →