TIFLUADOM, A KAPPA-OPIATE AGONIST, ACTS AS A PERIPHERAL CHOLECYSTOKININ RECEPTOR ANTAGONIST

被引：24

作者：

CHANG, RSL

LOTTI, VJ

CHEN, TB

KEEGAN, ME

机构：

来源：

NEUROSCIENCE LETTERS | 1986年 / 72卷 / 02期

关键词：

D O I：

10.1016/0304-3940(86)90082-0

中图分类号：

Q189 [神经科学];

学科分类号：

071006 ;

摘要：

引用

页码：211 / 214

页数：4

共 10 条

[1] BIOCHEMICAL AND PHARMACOLOGICAL CHARACTERIZATION OF AN EXTREMELY POTENT AND SELECTIVE NONPEPTIDE CHOLECYSTOKININ ANTAGONIST [J].

CHANG, RSL ;

LOTTI, VJ .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (13) :4923-4926

[2] A POTENT NONPEPTIDE CHOLECYSTOKININ ANTAGONIST SELECTIVE FOR PERIPHERAL-TISSUES ISOLATED FROM ASPERGILLUS-ALLIACEUS [J].

CHANG, RSL ;

LOTTI, VJ ;

MONAGHAN, RL ;

BIRNBAUM, J ;

STAPLEY, EO ;

GOETZ, MA ;

ALBERSSCHONBERG, G ;

PATCHETT, AA ;

LIESCH, JM ;

HENSENS, OD ;

SPRINGER, JP .

SCIENCE, 1985, 230 (4722) :177-179

[3] FURTHER EVIDENCE THAT SUBSTANCE-P PARTLY MEDIATES THE ACTION OF CHOLECYSTOKININ OCTAPEPTIDE (CCK-8) ON THE GUINEA-PIG ILEUM BUT NOT GALLBLADDER - STUDIES WITH A SUBSTANCE-P ANTAGONIST [J].

CHANG, RSL ;

LOTTI, VJ ;

CHEN, TB .

NEUROSCIENCE LETTERS, 1984, 46 (01) :71-75

[4] DESIGN OF POTENT, ORALLY EFFECTIVE, NONPEPTIDAL ANTAGONISTS OF THE PEPTIDE-HORMONE CHOLECYSTOKININ [J].

EVANS, BE ;

BOCK, MG ;

RITTLE, KE ;

DIPARDO, RM ;

WHITTER, WL ;

VEBER, DF ;

ANDERSON, PS ;

FREIDINGER, RM .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (13) :4918-4922

[5] PROGLUMIDE AND BENZOTRIPT - MEMBERS OF A DIFFERENT CLASS OF CHOLECYSTOKININ RECEPTOR ANTAGONISTS [J].

HAHNE, WF ;

JENSEN, RT ;

LEMP, GF ;

GARDNER, JD .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (10) :6304-6308

[6] REVERSE STEREOSELECTIVITY OF OPIATE AND BENZODIAZEPINE RECEPTORS FOR THE OPIOID BENZODIAZEPINE TIFLUADOM [J].

KLEY, H ;

SCHEIDEMANTEL, U ;

BERING, B ;

MULLER, WE .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 87 (04) :503-504

[7] THE EFFECT OF THE OPIOID-BENZODIAZEPINE, TIFLUADOM, ON INGESTIVE BEHAVIORS [J].

MORLEY, JE ;

LEVINE, AS ;

GRACE, M ;

KNEIP, J ;

ZEUGNER, H .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 93 (3-4) :265-269

[8] AN OPIOID BENZODIAZEPINE [J].

ROMER, D ;

BUSCHER, HH ;

HILL, RC ;

MAURER, R ;

PETCHER, TJ ;

ZEUGNER, H ;

BENSON, W ;

FINNER, E ;

MILKOWSKI, W ;

THIES, PW .

NATURE, 1982, 298 (5876) :759-760

[9]

SMITH GP, 1975, PHARMACOL BIOCHEM BE, V3, P135

[10] CHOLECYSTOKININ ANTAGONISTS SELECTIVELY POTENTIATE ANALGESIA INDUCED BY ENDOGENOUS OPIATES [J].

WATKINS, LR ;

KINSCHECK, IB ;

KAUFMAN, EFS ;

MILLER, J ;

FRENK, H ;

MAYER, DJ .

BRAIN RESEARCH, 1985, 327 (1-2) :181-190

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