AN EXPEDIENT ROUTE TO INDOLE-3-ACETIC-ACID DERIVATIVES

被引：0

作者：

SAMIZU, K ^{[1
]}

OGASAWARA, K ^{[1
]}

机构：

[1] TOHOKU UNIV,INST PHARMACEUT,SENDAI 98077,JAPAN

来源：

SYNLETT | 1994年 / 07期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An expedient synthesis of indole-3-acetic acid derivatives has been developed by employing the Heck reaction between 2-iodoaniline derivatives and 2,5-dihydro-dimethoxyfuran as the key step.

引用

页码：499 / 500

页数：2

共 5 条

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[5] CARBON-DIOXIDE - A REAGENT FOR THE SIMULTANEOUS PROTECTION OF NUCLEOPHILIC CENTERS AND THE ACTIVATION OF ALTERNATIVE LOCATIONS TO ELECTROPHILIC ATTACK - .3. A NEW SYNTHETIC METHOD FOR THE ORTHO-SUBSTITUTION OF N-MONOALKYLANILINES [J].

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