SYNTHESES AND ANTIFOLATE ACTIVITY OF 5-METHYL-5-DEAZA ANALOGS OF AMINOPTERIN, METHOTREXATE, FOLIC-ACID, AND N-10-METHYLFOLIC ACID

被引：118

作者：

PIPER, JR

MCCALEB, GS

MONTGOMERY, JA

KISLIUK, RL

GAUMONT, Y

SIROTNAK, FM

机构：

[1] TUFTS UNIV,SCH MED,DEPT BIOCHEM & PHARMACOL,BOSTON,MA 02111

[2] MEM SLOAN KETTERING CANC CTR,NEW YORK,NY 10021

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 06期

关键词：

D O I：

10.1021/jm00156a029

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1080 / 1087

页数：8

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