THE DISCOVERY OF SULFONAMIDE ENDOTHELIN ANTAGONISTS AND THE DEVELOPMENT OF THE ORALLY-ACTIVE ET(A) ANTAGONIST 5-(DIMETHYLAMINO)-N-(3,4-DIMETHYL-5-ISOXAZOLYL)-1-NAPHTHALENESULFONAMIDE

被引：141
作者：
STEIN, PD
HUNT, JT
FLOYD, DM
MORELAND, S
DICKINSON, KEJ
MITCHELL, C
LIU, ECK
WEBB, ML
MURUGESAN, N
DICKEY, J
MCMULLEN, D
ZHANG, RG
LEE, VG
SERAFINO, R
DELANEY, C
SCHAEFFER, TR
KOZLOWSKI, M
机构：
[1] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,DEPT CHEM CARDIOVASC AGENTS,PRINCETON,NJ 08543
[2] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,DEPT CARDIOVASC BIOCHEM,PRINCETON,NJ 08543
[3] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,DEPT PHARMACOL,PRINCETON,NJ 08543
[4] BRISTOL MYERS SQUIBB CO,PHARMACEUT RES INST,DEPT BIOMOLEC SCREENING,WALLINGFORD,CT 06492
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1994年 / 37卷 / 03期
关键词：
D O I：
10.1021/jm00029a001
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：329 / 331
页数：3
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