MUTAGENESIS OF THE BETA-2-ADRENERGIC RECEPTOR - HOW STRUCTURE ELUCIDATES FUNCTION

被引:107
作者
OSTROWSKI, J
KJELSBERG, MA
CARON, MG
LEFKOWITZ, RJ
机构
[1] DUKE UNIV, MED CTR, HOWARD HUGHES MED INST, DURHAM, NC 27710 USA
[2] DUKE UNIV, MED CTR, DEPT BIOCHEM, DURHAM, NC 27710 USA
[3] DUKE UNIV, MED CTR, DEPT CELL BIOL, DURHAM, NC 27710 USA
关键词
BETA-2-ADRENERGIC RECEPTOR; G-PROTEIN; MUTAGENESIS;
D O I
10.1146/annurev.pa.32.040192.001123
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:167 / 183
页数:17
相关论文
共 60 条
[1]   ISOPROTERENOL RESPONSE FOLLOWING TRANSFECTION OF THE MOUSE BETA-2-ADRENERGIC RECEPTOR GENE INTO Y1-CELLS [J].
ALLEN, JM ;
BAETGE, EE ;
ABRASS, IB ;
PALMITER, RD .
EMBO JOURNAL, 1988, 7 (01) :133-138
[2]   CYTOPLASMIC LOOP OF BETA-ADRENERGIC RECEPTORS - SYNAPTIC AND INTRACELLULAR-LOCALIZATION AND RELATION TO CATECHOLAMINERGIC NEURONS IN THE NUCLEI OF THE SOLITARY TRACTS [J].
AOKI, C ;
ZEMCIK, BA ;
STRADER, CD ;
PICKEL, VM .
BRAIN RESEARCH, 1989, 493 (02) :331-347
[3]   THE MAMMALIAN BETA-ADRENERGIC-RECEPTOR - STRUCTURAL AND FUNCTIONAL-CHARACTERIZATION OF THE CARBOHYDRATE MOIETY [J].
BENOVIC, JL ;
STANISZEWSKI, C ;
CERIONE, RA ;
CODINA, J ;
LEFKOWITZ, RJ ;
CARON, MG .
JOURNAL OF RECEPTOR RESEARCH, 1987, 7 (1-4) :257-281
[4]  
BEYER RM, 1990, EMBO J, V9, P2679
[5]  
BOEGE F, 1988, J BIOL CHEM, V263, P9040
[6]   PRIMARY STRUCTURE OF THE RAT BETA-2 ADRENERGIC-RECEPTOR GENE [J].
BUCKLAND, PR ;
HILL, RM ;
TIDMARSH, SF ;
MCGUFFIN, P .
NUCLEIC ACIDS RESEARCH, 1990, 18 (03) :682-682
[7]   SPECIFIC ACTIVATION OF GS BY SYNTHETIC PEPTIDES CORRESPONDING TO AN INTRACELLULAR LOOP OF THE BETA-ADRENERGIC-RECEPTOR [J].
CHEUNG, AH ;
HUANG, RRC ;
GRAZIANO, MP ;
STRADER, CD .
FEBS LETTERS, 1991, 279 (02) :277-280
[8]  
CHUNG FZ, 1988, J BIOL CHEM, V263, P4052
[9]  
COTECCHIA S, 1991, UNPUB DISCRETE AMINO
[10]   CLONING OF THE GENE AND CDNA FOR MAMMALIAN BETA-ADRENERGIC-RECEPTOR AND HOMOLOGY WITH RHODOPSIN [J].
DIXON, RAF ;
KOBILKA, BK ;
STRADER, DJ ;
BENOVIC, JL ;
DOHLMAN, HG ;
FRIELLE, T ;
BOLANOWSKI, MA ;
BENNETT, CD ;
RANDS, E ;
DIEHL, RE ;
MUMFORD, RA ;
SLATER, EE ;
SIGAL, IS ;
CARON, MG ;
LEFKOWITZ, RJ ;
STRADER, CD .
NATURE, 1986, 321 (6065) :75-79