REVERSE PHARMACOLOGY OF THE NICOTINIC ACETYLCHOLINE-RECEPTOR - MAPPING THE LOCAL-ANESTHETIC BINDING-SITE

被引:23
作者
LEONARD, RJ [1 ]
CHARNET, P [1 ]
LABARCA, C [1 ]
VOGELAAR, NJ [1 ]
CZYZYK, L [1 ]
GOUIN, A [1 ]
DAVIDSON, N [1 ]
LESTER, HA [1 ]
机构
[1] CALTECH,DEPT BIOL,PASADENA,CA 91125
关键词
D O I
10.1111/j.1749-6632.1991.tb33894.x
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
[No abstract available]
引用
收藏
页码:588 / 599
页数:12
相关论文
共 29 条
[1]   VOLTAGE JUMP ANALYSIS OF PROCAINE ACTION AT FROG ENDPLATE [J].
ADAMS, PR .
JOURNAL OF PHYSIOLOGY-LONDON, 1977, 268 (02) :291-318
[2]   MOLECULAR-CLONING OF CDNA CODING FOR THE GAMMA-SUBUNIT OF TORPEDO ACETYLCHOLINE-RECEPTOR [J].
BALLIVET, M ;
PATRICK, J ;
LEE, J ;
HEINEMANN, S .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1982, 79 (14) :4466-4470
[3]  
BOULTER J, 1985, J NEUROSCI, V5, P2545
[4]   ISOLATION AND SEQUENCE OF CDNA CLONES CODING FOR THE PRECURSOR TO THE GAMMA-SUBUNIT OF MOUSE MUSCLE NICOTINIC ACETYLCHOLINE-RECEPTOR [J].
BOULTER, J ;
EVANS, K ;
MARTIN, G ;
MASON, P ;
STENGELIN, S ;
GOLDMAN, D ;
HEINEMANN, S ;
PATRICK, J .
JOURNAL OF NEUROSCIENCE RESEARCH, 1986, 16 (01) :37-49
[5]   EFFECTS OF CHLORPROMAZINE AND PHENCYCLIDINE ON MOUSE C2 ACETYLCHOLINE-RECEPTOR KINETICS [J].
CHANGEUX, JP ;
PINSET, C ;
RIBERA, AB .
JOURNAL OF PHYSIOLOGY-LONDON, 1986, 378 :497-513
[6]   AN OPEN-CHANNEL BLOCKER INTERACTS WITH ADJACENT TURNS OF ALPHA-HELICES IN THE NICOTINIC ACETYLCHOLINE-RECEPTOR [J].
CHARNET, P ;
LABARCA, C ;
LEONARD, RJ ;
VOGELAAR, NJ ;
CZYZYK, L ;
GOUIN, A ;
DAVIDSON, N ;
LESTER, HA .
NEURON, 1990, 4 (01) :87-95
[7]   NUCLEOTIDE AND DEDUCED AMINO-ACID-SEQUENCES OF TORPEDO-CALIFORNICA ACETYLCHOLINE-RECEPTOR GAMMA-SUBUNIT [J].
CLAUDIO, T ;
BALLIVET, M ;
PATRICK, J ;
HEINEMANN, S .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (04) :1111-1115
[8]  
COURTNEY KR, 1987, HDB EXPT PHARM, V81, pCH3
[9]   COMPLETE MESSENGER-RNA CODING SEQUENCE OF THE ACETYLCHOLINE BINDING ALPHA-SUBUNIT OF TORPEDO-MARMORATA ACETYLCHOLINE-RECEPTOR - A MODEL FOR THE TRANSMEMBRANE ORGANIZATION OF THE POLYPEPTIDE-CHAIN [J].
DEVILLERSTHIERY, A ;
GIRAUDAT, J ;
BENTABOULET, M ;
CHANGEUX, JP .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (07) :2067-2071
[10]   STRUCTURE OF THE HIGH-AFFINITY BINDING-SITE FOR NONCOMPETITIVE BLOCKERS OF THE ACETYLCHOLINE-RECEPTOR - SERINE-262 OF THE DELTA-SUBUNIT IS LABELED BY [H-3] CHLORPROMAZINE [J].
GIRAUDAT, J ;
DENNIS, M ;
HEIDMANN, T ;
CHANG, JY ;
CHANGEUX, JP .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (08) :2719-2723