ENKEPHALINASE - SELECTIVE PEPTIDE INHIBITORS

被引:151
作者
HUDGIN, RL
CHARLESON, SE
ZIMMERMAN, M
MUMFORD, R
WOOD, PL
机构
[1] MERCK FROSST LABS,DEPT PHARMACOL,POINTE CLAIRE H9R 4D8,QUEBEC,CANADA
[2] MERCK SHARP & DOHME,DEPT IMMUNOL,RAHWAY,NJ 07065
关键词
D O I
10.1016/0024-3205(81)90632-9
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2593 / 2601
页数:9
相关论文
共 33 条
[1]   SEPARATION OF HUMAN-BRAIN ANGIOTENSIN-CONVERTING ENZYME FROM ENKEPHALIN-DEGRADING ACTIVITY [J].
ARREGUI, A ;
LEE, CM ;
EMSON, PC ;
IVERSEN, LL .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 59 (1-2) :141-144
[2]   INHIBITION OF ENKEPHALIN-DEGRADING AMINOPEPTIDASE ACTIVITY BY CERTAIN PEPTIDES [J].
BARCLAY, RK ;
PHILLIPPS, MA .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 96 (04) :1732-1738
[3]   CO-IDENTITY OF BRAIN ANGIOTENSIN CONVERTING ENZYME WITH A MEMBRANE-BOUND DIPEPTIDYL CARBOXYPEPTIDASE INACTIVATING MET - ENKEPHALIN [J].
BENUCK, M ;
MARKS, N .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1979, 88 (01) :215-221
[4]   CHARACTERIZATION OF A DISTINCT MEMBRANE-BOUND DIPEPTIDYL CARBOXYPEPTIDASE INACTIVATING ENKEPHALIN IN BRAIN [J].
BENUCK, M ;
MARKS, N .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 95 (02) :822-828
[5]  
CLELAND WW, 1967, ADV ENZYMOL RAMB, V29, P1
[6]  
CRAVES FB, 1978, J PHARMACOL EXP THER, V206, P492
[7]   SPECTROPHOTOMETRIC ASSAY AND PROPERTIES OF ANGIOTENSIN-CONVERTING ENZYME OF RABBIT LUNG [J].
CUSHMAN, DW ;
CHEUNG, HS .
BIOCHEMICAL PHARMACOLOGY, 1971, 20 (07) :1637-+
[8]   EXTREMELY RAPID DEGRADATION OF [H-3] METHIONINE-ENKEPHALIN BY VARIOUS RAT TISSUES INVIVO AND INVITRO [J].
DUPONT, A ;
CUSAN, L ;
GARON, M ;
ALVARADOURBINA, G ;
LABRIE, F .
LIFE SCIENCES, 1977, 21 (07) :907-914
[9]   2 DISTINCT ENKEPHALINASES - SOLUBILIZATION, PARTIAL-PURIFICATION AND SEPARATION FROM ANGIOTENSIN CONVERTING ENZYME [J].
GORENSTEIN, C ;
SNYDER, SH .
LIFE SCIENCES, 1979, 25 (24-2) :2065-2070
[10]   ISOLATION OF AN ENDOGENOUS COMPOUND FROM BRAIN WITH PHARMACOLOGICAL PROPERTIES SIMILAR TO MORPHINE [J].
HUGHES, J .
BRAIN RESEARCH, 1975, 88 (02) :295-308