MORPHINE ANALGESIA AFTER INTRATHECAL ADMINISTRATION OF A NARCOTIC AGONIST, CHLOROXYMORPHAMINE AND ANTAGONIST, CHLORNALTREXAMINE

被引:9
作者
LARSON, AA
ARMSTRONG, MJ
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关键词
D O I
10.1016/0014-2999(80)90056-4
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:25 / 31
页数:7
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共 13 条
[1]   CHLOROXYMORPHAMINE, AN OPIOID RECEPTOR SITE-DIRECTED ALKYLATING AGENT HAVING NARCOTIC AGONIST ACTIVITY [J].
CARUSO, TP ;
TAKEMORI, AE ;
LARSON, DL ;
PORTOGHESE, PS .
SCIENCE, 1979, 204 (4390) :316-318
[2]  
CARUSO TP, 1979, FED PROC, V38, P1894
[3]  
CARUSO TP, J PHARMACOL EXP THER
[4]  
D'amour FE, 1941, J PHARMACOL EXP THER, V72, P74
[5]  
LITCHFIELD JT, 1949, J PHARMACOL EXP THER, V96, P99
[6]   SYNTHESIS AND PHARMACOLOGIC CHARACTERIZATION OF AN ALKYLATING ANALOG (CHLORNALTREXAMINE) OF NALTREXONE WITH ULTRA-LONG-LASTING NARCOTIC-ANTAGONIST PROPERTIES [J].
PORTOGHESE, PS ;
LARSON, DL ;
JIANG, JB ;
CARUSO, TP ;
TAKEMORI, AE .
JOURNAL OF MEDICINAL CHEMISTRY, 1979, 22 (02) :168-173
[7]   6-BETA [N,N-BIS(2-CHLOROETHYL)AMINO]-17-(CYCLOPROPYLMETHYL)-4,5-ALPHA-EPOXY-3,14-DIHYDROXYMORPHINAN (CHLORANALTREXAMINE) - POTENT OPIOID RECEPTOR ALKYLATING AGENT WITH ULTRALONG NARCOTIC-ANTAGONIST ACTIVITY [J].
PORTOGHESE, PS ;
LARSON, DL ;
JIANG, JB ;
TAKEMORI, AE ;
CARUSO, TP .
JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (07) :598-599
[8]   ANTINOCICEPTIVE EFFECT OF INTRATHECALLY ADMINISTERED SEROTONIN [J].
WANG, JK .
ANESTHESIOLOGY, 1977, 47 (03) :269-271
[9]  
YAKSH TL, 1979, J PHARMACOL EXP THER, V208, P446
[10]   NARCOTIC ANALGETICS - CNS SITES AND MECHANISMS OF ACTION AS REVEALED BY INTRA-CEREBRAL INJECTION TECHNIQUES [J].
YAKSH, TL ;
RUDY, TA .
PAIN, 1978, 4 (04) :299-359