FACILE INTRAMOLECULAR CYCLOADDITIONS OF 2-(N-ACYLAMINO)-1-THIA-1,3-DIENES

被引：9

作者：

BARNISH, IT

FISHWICK, CWG

HILL, DR

机构：

[1] UNIV LEEDS,SCH CHEM,LEEDS LS2 9JT,W YORKSHIRE,ENGLAND

[2] PFIZER LTD,SANDWICH CT13 9NJ,KENT,ENGLAND

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 03期

关键词：

D O I：

10.1016/S0040-4039(00)92640-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

2-(N-Acylamino)-1-thia-1,3-dienes, generated via acylation of readily available alpha,beta-unsaturated thioamides, undergo regio- and stereospecific intramolecular Diels-Alder cycloaddition with unactivated olefinic and acetylenic dienophiles to yield polycyclic dihydrothiopyrans.

引用

页码：405 / 408

页数：4

共 50 条

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