STUDIES ON THE CHEMISTRY OF THIENOANELLATED O,N-CONTAINING AND S,N-CONTAINING HETEROCYCLES .6. SYNTHESIS OF SOME THIENOANELLATED [1,4]BENZOXAZEPINES

被引：3

作者：

LAIMER, I

ERKER, T

机构：

[1] Institute of Pharmaceutical Chemistry, University of Vienna, Vienna, A-1090

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1994年 / 31卷 / 04期

关键词：

D O I：

10.1002/jhet.5570310460

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Substituted thieno[2,3-b][1,4]benzoxazepine derivatives as well as thieno[3,2-b][1,4]benzoxazepine derivatives have been synthesized. They are thienoanalogues of loxapine, a potent antipsychotic drug. Research activities concentrate on the preparation of structurally modified compounds of loxapine to minimize its undesirable extrapyramidal symptoms.

引用

页码：1053 / 1059

页数：7

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