IRREVERSIBLE ENZYME INHIBITORS .115. PROTEOLYTIC ENZYMES .5. ACTIVE-SITE-DIRECTED IRREVERSIBLE INHIBITORS OF TRYPSIN DERIVED FROM P-(PHENOXYALKOXY)BENZAMIDINES WITH A TERMINAL SULFONYL FLUORIDE

被引：44

作者：

BAKER, BR

ERICKSON, EH

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1968年 / 11卷 / 02期

关键词：

D O I：

10.1021/jm00308a011

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：245 / &

共 17 条

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[2] IRREVERSIBLE ENZYME INHIBITORS .114. PROTEOLYTIC ENZYMES .4. ADDITIONAL ACTIVE-SITE-DIRECTED IRREVERSIBLE INHIBITORS OF ALPHA-CHYMOTRYPSIN DERIVED FROM PHENOXYACETAMIDES BEARING A TERMINAL SULFONYL FLUORIDE [J].

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[3] IRREVERSIBLE ENZYME INHIBITORS .106. PROTEOLYTIC ENZYMES .I. BULK TOLERANCES IN TRYPSIN-INHIBITOR COMPLEXES [J].

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[4] ANALOGS OF TETRAHYDROFOLIC ACID .39(1,2). SELECTIVE BROMOACYLATION OF POLYFUNCTIONAL MOLECULES FOR SYNTHESIS OF ACTIVE-SITE-DIRECTED IRREVERSIBLE ENZYME INHIBITORS [J].

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[10] PREPARATION AND PROPERTIES OF 2 NEW CHROMOGENIC SUBSTRATES OF TRYPSIN [J].

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