BIFUNCTIONAL CHIRAL AUXILIARIES .2. THE SYNTHESIS OF 1,3-DIACYLIMIDAZOLIDIN-2-ONES FROM 1,2-DIAMINES

被引：37

作者：

DAVIES, SG

MORTLOCK, AA

机构：

[1] The Dyson Perrins Laboratory, Oxford, OX1 3QY, South Parks Road

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 36期

关键词：

D O I：

10.1016/S0040-4039(00)92309-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The title compounds are readily prepared in three steps via the corresponding 1,3-diacylimidazolidine-2-thiones. The final step involves the novel use of mercury (II) acetate for the conversion of thioureas to ureas.

引用

页码：4791 / 4794

页数：4

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