AZELASTINE INHIBITS BRONCHIAL HYPERREACTIVITY TO ACETYLCHOLINE IN GUINEA-PIGS

被引:6
作者
ACHTERRATHTUCKERMANN, U [1 ]
SZELENYI, I [1 ]
机构
[1] ASTA PHARMA AG,DEPT PHARMACOL,POB 100503,D-6000 FRANKFURT MAIN 1,FED REP GER
来源
EXPERIENTIA | 1988年 / 44卷 / 11-12期
关键词
D O I
10.1007/BF01939898
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:993 / 996
页数:4
相关论文
共 22 条
[1]   AZELASTINE, A NEW ANTIALLERGIC ANTIASTHMATIC AGENT, INHIBITS PAF-ACETHER-INDUCED PLATELET-AGGREGATION, PAW EDEMA AND BRONCHOCONSTRICTION [J].
ACHTERRATHTUCKERMANN, U ;
WEISCHER, CH ;
SZELENYI, I .
PHARMACOLOGY, 1988, 36 (04) :265-271
[2]   INHIBITION OF CYSTEINYL-LEUKOTRIENE PRODUCTION BY AZELASTINE AND ITS BIOLOGICAL SIGNIFICANCE [J].
ACHTERRATHTUCKERMANN, U ;
SIMMET, T ;
LUCK, W ;
SZELENYI, I ;
PESKAR, BA .
AGENTS AND ACTIONS, 1988, 24 (3-4) :217-223
[3]  
BOULET LP, 1984, AM REV RESPIR DIS, V130, P368
[4]   ALLERGEN-INDUCED INCREASE IN BRONCHIAL RESPONSIVENESS TO HISTAMINE - RELATIONSHIP TO THE LATE ASTHMATIC RESPONSE AND CHANGE IN AIRWAY CALIBER [J].
CARTIER, A ;
THOMSON, NC ;
FRITH, PA ;
ROBERTS, R ;
HARGREAVE, FE .
JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY, 1982, 70 (03) :170-177
[5]   ANTAGONISM OF HISTAMINE AND LEUKOTRIENES BY AZELASTINE IN ISOLATED GUINEA-PIG ILEUM [J].
CHAND, N ;
DIAMANTIS, W ;
SOFIA, RD .
AGENTS AND ACTIONS, 1986, 19 (3-4) :164-168
[6]   INHIBITION OF LEUKOTRIENE (SRS-A)-MEDIATED ACUTE LUNG ANAPHYLAXIS BY AZELASTINE IN GUINEA-PIGS [J].
CHAND, N ;
NOLAN, K ;
DIAMANTIS, W ;
PERHACH, JL ;
SOFIA, RD .
ALLERGY, 1986, 41 (07) :473-478
[7]   INHIBITION OF PASSIVE CUTANEOUS ANAPHYLAXIS (PCA) BY AZELASTINE - DISSOCIATION OF ITS ANTIALLERGIC ACTIVITIES FROM ANTIHISTAMINIC AND ANTISEROTONIN PROPERTIES [J].
CHAND, N ;
HARRISON, JE ;
ROONEY, SM ;
SOFIA, RD ;
DIAMANTIS, W .
INTERNATIONAL JOURNAL OF IMMUNOPHARMACOLOGY, 1985, 7 (06) :833-838
[8]   INHIBITION OF IGE-MEDIATED ALLERGIC HISTAMINE-RELEASE FROM RAT PERITONEAL MAST-CELLS BY AZELASTINE AND SELECTED ANTIALLERGIC DRUGS [J].
CHAND, N ;
PILLAR, J ;
DIAMANTIS, W ;
SOFIA, RD .
AGENTS AND ACTIONS, 1985, 16 (05) :318-322
[9]   SPIRALLY CUT TRACHEAL STRIP PREPARATION [J].
CONSTANTINE, JW .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1965, 17 (06) :384-+
[10]  
CUSS FM, 1986, LANCET, V2, P189