EXPERIMENTS ON THE MODE OF ACTION OF PIRIPROST (U-60,257), AN INHIBITOR OF LEUKOTRIENE FORMATION IN CLONED MOUSE MAST-CELLS AND IN RAT BASOPHIL LEUKEMIA-CELLS

被引:16
作者
BACH, MK
BRASHLER, JR
WHITE, GJ
GALLI, SJ
机构
[1] UPJOHN CO, DEPT HYPERSENSITIV DIS RES, KALAMAZOO, MI 49001 USA
[2] BETH ISRAEL HOSP, DEPT PATHOL, BOSTON, MA 02215 USA
[3] HARVARD UNIV, SCH MED, BOSTON, MA 02115 USA
[4] BETH ISRAEL HOSP, CHARLES A DANA RES INST, BOSTON, MA 02215 USA
关键词
D O I
10.1016/0006-2952(87)90111-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1461 / 1466
页数:6
相关论文
共 27 条
[1]   PROSPECTS FOR THE INHIBITION OF LEUKOTRIENE SYNTHESIS [J].
BACH, MK .
BIOCHEMICAL PHARMACOLOGY, 1984, 33 (04) :515-521
[3]   SOLUBILIZATION AND CHARACTERIZATION OF THE LEUKOTRIENE-C4 SYNTHETASE OF RAT BASOPHIL LEUKEMIA-CELLS - A NOVEL, PARTICULATE GLUTATHIONE S-TRANSFERASE [J].
BACH, MK ;
BRASHLER, JR ;
MORTON, DR .
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1984, 230 (02) :455-465
[4]  
BACH MK, 1982, PROSTAGLANDINS, V23, P759
[5]   LEUKOTRIENE-C SYNTHETASE, A SPECIAL GLUTATHIONE S-TRANSFERASE - PROPERTIES OF THE ENZYME AND INHIBITOR STUDIES WITH SPECIAL REFERENCE TO THE MODE OF ACTION OF U-60,257, A SELECTIVE INHIBITOR OF LEUKOTRIENE SYNTHESIS [J].
BACH, MK ;
BRASHLER, JR ;
PECK, RE ;
MORTON, DR .
JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY, 1984, 74 (03) :353-357
[6]  
BACH MK, 1985, RES COMMUN CHEM PATH, V49, P361
[7]   PHARMACOLOGICAL MODULATION OF HUMAN EOSINOPHIL LEUKOTRIENE-C4 PRODUCTION [J].
CROMWELL, O ;
SHAW, RJ ;
KAY, AB .
PROSTAGLANDINS, 1984, 28 (05) :654-654
[8]   ALLERGEN CHALLENGE OF LUNG-TISSUE FROM ASTHMATICS ELICITS BRONCHIAL CONTRACTION THAT CORRELATES WITH THE RELEASE OF LEUKOTRIENE-C4, LEUKOTRIENE-D4, AND LEUKOTRIENE-E4 [J].
DAHLEN, SE ;
HANSSON, G ;
HEDQVIST, P ;
BJORCK, T ;
GRANSTROM, E ;
DAHLEN, B .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (06) :1712-1716
[9]   MAST-CELL CLONES - A MODEL FOR THE ANALYSIS OF CELLULAR MATURATION [J].
GALLI, SJ ;
DVORAK, AM ;
MARCUM, JA ;
ISHIZAKA, T ;
NABEL, G ;
DERSIMONIAN, H ;
PYNE, K ;
GOLDIN, JM ;
ROSENBERG, RD ;
CANTOR, H ;
DVORAK, HF .
JOURNAL OF CELL BIOLOGY, 1982, 95 (02) :435-444
[10]  
GALLI SJ, 1985, CELL IMMUNOL, V22, P233