SYNTHESIS AND BIOLOGICAL PROPERTIES OF ENKEPHALIN-LIKE PEPTIDES CONTAINING CARBORANYLALANINE IN PLACE OF PHENYLALANINE

被引：26
作者：
SCHWYZER, R
DO, KQ
EBERLE, AN
FAUCHERE, JL
机构：
来源：
HELVETICA CHIMICA ACTA | 1981年 / 64卷 / 07期
关键词：
D O I：
10.1002/hlca.19810640712
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
引用
收藏
页码：2078 / 2083
页数：6
相关论文
共 29 条
[1]   OXIDATIVE REACTIONS OF HYDRAZINES .2. ISOPHTHALIMIDES - NEW PROTECTIVE GROUPS ON NITROGEN [J].
CARPINO, LA .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1957, 79 (01) :98-101
[2]  
CASTELL JV, 1979, HELV CHIM ACTA, V62, P525, DOI 10.1002/hlca.19790620219
[3]   SYNTHESIS AND OPIOID ACTIVITIES OF STEREOISOMERS AND OTHER D-AMINO-ACID ANALOGS OF METHIONINE-ENKEPHALIN [J].
COY, DH ;
KASTIN, AJ ;
SCHALLY, AV ;
MORIN, O ;
CARON, NG ;
LABRIE, F ;
WALKER, JM ;
FERTEL, R ;
BERNTSON, GG ;
SANDMAN, CA .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1976, 73 (03) :632-638
[4]   SYNTHESIS OF (S)-(+)-2-AMINO-3-(1-ADAMANTYL)-PROPIONIC ACID (L-(+)-ADAMANTYLALANINE,ADA) AS A FAT OR SUPER ANALOG OF LEUCINE AND PHENYLALANINE [J].
DO, KQ ;
THANEI, P ;
CAVIEZEL, M ;
SCHWYZER, R .
HELVETICA CHIMICA ACTA, 1979, 62 (04) :956-964
[5]   SYNTHESIS AND BIOLOGICAL PROPERTIES OF ENKEPHALIN-LIKE PEPTIDES CONTAINING ADAMANTYLALANINE IN POSITION 4 AND 5 [J].
DO, KQ ;
SCHWYZER, R .
HELVETICA CHIMICA ACTA, 1981, 64 (07) :2084-2089
[6]   ELECTRONIC, STERIC, AND HYDROPHOBIC FACTORS INFLUENCING THE ACTION OF ENKEPHALIN-LIKE PEPTIDES ON OPIATE RECEPTORS [J].
DO, KQ ;
FAUCHERE, JL ;
SCHWYZER, R ;
SCHILLER, PW ;
LEMIEUX, C .
HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 1981, 362 (06) :601-610
[7]  
DO KQ, 1980, THESIS EPFZ
[8]   HORMONE-RECEPTOR INTERACTIONS - [4-CARBORANYLALANINE, 5-LEUCINE]-ENKEPHALIN AS A STRUCTURAL PROBE FOR OPIATE RECEPTOR [J].
EBERLE, A ;
LEUKART, O ;
SCHILLER, P ;
FAUCHERE, J ;
SCHWYZER, R .
FEBS LETTERS, 1977, 82 (02) :325-328
[9]   SYNTHESIS, ENZYMIC DEGRADATION, LIPOPHILIC PROPERTIES, AND BIOLOGICAL-ACTIVITY OF [D-ALANINE2, TERT-BUTYLGLYCINE5]ENKEPHALIN AMIDE [J].
FAUCHERE, JL ;
PETERMANN, C .
HELVETICA CHIMICA ACTA, 1980, 63 (04) :824-831
[10]   SYNTHESIS OF [4-CARBORANYLALANINE, 5-LEUCINE]-ENKEPHALIN - (INCLUDING AN IMPROVED PREPARATION OF TERT-BUTOXYCARBONYL-L-ORTHO-CARBORANYLALANINE, NEW DERIVATIVES OF L-PROPARGYLGLYCINE, AND A NOTE ON MELANOTROPIC AND OPIATE RECEPTOR-BINDING CHARACTERISTICS) [J].
FAUCHERE, JL ;
LEUKART, O ;
EBERLE, A ;
SCHWYZER, R .
HELVETICA CHIMICA ACTA, 1979, 62 (05) :1385-1395
123