7-CHLOROKYNURENIC ACID IS A SELECTIVE ANTAGONIST AT THE GLYCINE MODULATORY SITE OF THE N-METHYL-D-ASPARTATE RECEPTOR COMPLEX

被引:577
作者
KEMP, JA
FOSTER, AC
LEESON, PD
PRIESTLEY, T
TRIDGETT, R
IVERSEN, LL
WOODRUFF, GN
机构
关键词
D O I
10.1073/pnas.85.17.6547
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
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页码:6547 / 6550
页数:4
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[1]   BIOCHEMICAL-EVIDENCE THAT GLYCINE ALLOSTERICALLY REGULATES AN NMDA RECEPTOR-COUPLED ION CHANNEL [J].
BONHAUS, DW ;
BURGE, BC ;
MCNAMARA, JO .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 142 (03) :489-490
[2]   INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
SCHMIECHEN, R ;
NEEF, G ;
NIELSEN, M ;
PETERSEN, EN .
SCIENCE, 1982, 216 (4551) :1241-1243
[3]   LIGHT MICROSCOPIC AUTORADIOGRAPHIC LOCALIZATION OF [H-3] GLYCINE AND [H-3] STRYCHNINE BINDING-SITES IN RAT-BRAIN [J].
BRISTOW, DR ;
BOWERY, NG ;
WOODRUFF, GN .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 126 (03) :303-307
[4]   CPP, A NEW POTENT AND SELECTIVE NMDA ANTAGONIST - DEPRESSION OF CENTRAL NEURON RESPONSES, AFFINITY FOR [H-3] D-AP5 BINDING-SITES ON BRAIN MEMBRANES AND ANTICONVULSANT ACTIVITY [J].
DAVIES, J ;
EVANS, RH ;
HERRLING, PL ;
JONES, AW ;
OLVERMAN, HJ ;
POOK, P ;
WATKINS, JC .
BRAIN RESEARCH, 1986, 382 (01) :169-173
[5]   A COMPARISON OF EXCITATORY AMINO-ACID ANTAGONISTS ACTING AT PRIMARY AFFERENT C-FIBERS AND MOTONEURONS OF THE ISOLATED SPINAL-CORD OF THE RAT [J].
EVANS, RH ;
EVANS, SJ ;
POOK, PC ;
SUNTER, DC .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 91 (03) :531-537
[6]   COMPARISON OF L-[H-3]GLUTAMATE, D-[H-3]ASPARTATE, DL-[H-3]AP5 AND [H-3] NMDA AS LIGANDS FOR NMDA RECEPTORS IN CRUDE POSTSYNAPTIC DENSITIES FROM RAT-BRAIN [J].
FOSTER, AC ;
FAGG, GE .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 133 (03) :291-300
[7]   IMPROVED PATCH-CLAMP TECHNIQUES FOR HIGH-RESOLUTION CURRENT RECORDING FROM CELLS AND CELL-FREE MEMBRANE PATCHES [J].
HAMILL, OP ;
MARTY, A ;
NEHER, E ;
SAKMANN, B ;
SIGWORTH, FJ .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1981, 391 (02) :85-100
[8]   COMPLEX STRUCTURE OF QUISQUALATE-SENSITIVE GLUTAMATE RECEPTORS IN RAT CORTEX [J].
HONORE, T ;
NIELSEN, M .
NEUROSCIENCE LETTERS, 1985, 54 (01) :27-32
[9]   GLYCINE POTENTIATES THE NMDA RESPONSE IN CULTURED MOUSE-BRAIN NEURONS [J].
JOHNSON, JW ;
ASCHER, P .
NATURE, 1987, 325 (6104) :529-531
[10]   ENHANCED SURVIVAL OF RAT NEONATAL CEREBRAL CORTICAL-NEURONS AT SUBATMOSPHERIC OXYGEN-TENSIONS INVITRO [J].
KAPLAN, FS ;
BRIGHTON, CT ;
BOYTIM, MJ ;
SELZER, ME ;
LEE, V ;
SPINDLER, K ;
SILBERBERG, D ;
BLACK, J .
BRAIN RESEARCH, 1986, 384 (01) :199-203