REACTIVATION BY CYSTEAMINE OF VASCULAR ALPHA-ADRENOCEPTORS BLOCKED BY THE TETRAMINE DISULFIDE BENEXTRAMINE AND INTERACTION OF BENEXTRAMINE WITH PHENOXYBENZAMINE

被引:8
作者
BRASILI, L
MELCHIORRE, C
BELLEAU, B
BENFEY, BG
机构
[1] MCGILL UNIV,DEPT PHARMACOL & THERAPEUT,MONTREAL H3G 1Y6,QUEBEC,CANADA
[2] MCGILL UNIV,DEPT CHEM,MONTREAL H3G 1Y6,QUEBEC,CANADA
关键词
D O I
10.1139/y80-224
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1490 / 1493
页数:4
相关论文
共 9 条
[1]  
BENFEY BG, 1980, FED PROC, V39, P1106
[2]   ANTAGONISM OF NOREPINEPHRINE RESPONSES OF ISOLATED RABBIT AORTA BY ALIPHATIC SULFUR-CONTAINING AMINES [J].
DEMAREE, GE ;
BROCKENTON, RE ;
HEIFFER, MH ;
ROTHE, WE .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1971, 60 (11) :1743-+
[3]  
FURCHGOTT RF, 1955, PHARMACOL REV, V7, P183
[4]  
Furchgott RF, 1966, ADV DRUG RES, P21
[5]  
GRAHAM JDP, 1962, PROGRESS MEDICINAL C, V2, P132
[6]  
HARVEY SC, 1954, J PHARMACOL EXP THER, V112, P274
[7]  
LIPPERT B, 1973, FRONTIERS CATECHOLAM, P369
[8]   MOLECULAR-PROPERTIES OF ADRENERGIC ALPHA-RECEPTOR .2. OPTIMUM COVALENT INHIBITION BY 2 DIFFERENT PROTOTYPES OF POLYAMINE DISULFIDES [J].
MELCHIORRE, C ;
YONG, MS ;
BENFEY, BG ;
BELLEAU, B .
JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (11) :1126-1132
[9]   MODIFICATION OF RECEPTOR THEORY [J].
STEPHENSON, RP .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1956, 11 (04) :379-393