SYNTHESIS OF A CONFORMATIONALLY CONSTRAINED ANALOG OF BW A78U, AN ANTICONVULSANT ADENINE DERIVATIVE

被引：14

作者：

DESAUBRY, L ^{[1
]}

WERMUTH, CG ^{[1
]}

BOURGUIGNON, JJ ^{[1
]}

机构：

[1] CTR NEUROCHIM,PHARMACOCHIM MOLEC LAB,CNRS,UPR 421,F-67084 STRASBOURG,FRANCE

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 24期

关键词：

D O I：

10.1016/0040-4039(95)00734-T

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of a conformationally constrained analogue of the anticonvulsant BW A78U, a 9-benzyl-adenine derivative, has been devised using silicon tetrachloride in a new cyclodehydration.

引用

页码：4249 / 4252

页数：4

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