PLASMA-CONCENTRATIONS AND PROTEIN-BINDING OF DISOPYRAMIDE AND MONO-N-DEALKYLDISOPYRAMIDE DURING CHRONIC ORAL DISOPYRAMIDE THERAPY

被引:38
作者
AITIO, ML
机构
[1] UNIV TURKU,DEPT PHARMACOL,SF-20500 TURKU 50,FINLAND
[2] UNIV HELSINKI,DEPT CLIN PHARMACOL,SF-00170 HELSINKI 17,FINLAND
[3] UNIV TURKU,DEPT MED,SF-20500 TURKU 50,FINLAND
关键词
D O I
10.1111/j.1365-2125.1981.tb01134.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:369 / 375
页数:7
相关论文
共 22 条
[1]   SIMULTANEOUS DETERMINATION OF DISOPYRAMIDE AND ITS MONO-N-DEALKYLATED METABOLITE IN PLASMA BY GAS-LIQUID-CHROMATOGRAPHY [J].
AITIO, ML .
JOURNAL OF CHROMATOGRAPHY, 1979, 164 (04) :515-520
[2]  
AITIO ML, 1979, ARCH INT PHARMACOD T, V239, P16
[3]   ENHANCED METABOLISM AND DIMINISHED EFFICACY OF DISOPYRAMIDE BY ENZYME-INDUCTION [J].
AITIO, ML ;
VUORENMAA, T .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 9 (02) :149-152
[4]  
AITIO ML, BRIT J CLIN PHARMAC
[5]  
BAINES MW, 1976, J INT MED RES, V4, P5
[6]  
Bazett HC, 1920, HEART-J STUD CIRC, V7, P353
[7]   DISOPYRAMIDE SERUM AND PHARMACOLOGIC EFFECT KINETICS APPLIED TO ASSESSMENT OF BIOAVAILABILITY [J].
BRYSON, SM ;
WHITING, B ;
LAWRENCE, JR .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1978, 6 (05) :409-419
[8]   COMPARATIVE BINDING OF DISOPYRAMIDE PHOSPHATE AND QUINIDINE SULFATE TO HUMAN PLASMA-PROTEINS [J].
CHIEN, YW ;
LAMBERT, HJ ;
KARIM, A .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1974, 63 (12) :1877-1879
[9]   SOME EFFECTS OF DISOPYRAMIDE AND ITS N-DE-ALKYLATED METABOLITE ON ISOLATED NERVE AND CARDIAC-MUSCLE [J].
GRANT, AM ;
MARSHALL, RJ ;
ANKIER, SI .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 49 (04) :389-394
[10]   DISOPYRAMIDE - REVIEW OF ITS PHARMACOLOGICAL PROPERTIES AND THERAPEUTIC USE IN TREATING CARDIAC-ARRHYTHMIAS [J].
HEEL, RC ;
BROGDEN, RN ;
SPEIGHT, TM ;
AVERY, GS .
DRUGS, 1978, 15 (05) :331-368